SCHEMBL2175829

SCHEMBL2175829

NC(=O)Nc1ccccc1Cl

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.75
KDM4E B2RXH2 4/20 0.65
HPGD P15428 1/20 0.62
CYP2C19 P33261 1/20 0.62
MEN1 O00255 4/20 0.60
KMT2A Q03164 4/20 0.60
MAPT P10636 3/20 0.57
LMNA P02545 2/20 0.57
ALDH1A1 P00352 2/20 0.57
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
GAA P10253 2/20 0.53
POLB P06746 2/20 0.53
HTT P42858 2/20 0.53
TAS1R3 Q7RTX0 1/20 0.53
TAS1R1 Q7RTX1 1/20 0.53
TAS1R2 Q8TE23 1/20 0.53
CASP3 P42574 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29537172 1.00 CYP1A2 (0.75) CYP1A2KDM4EHPGDCYP2C19MEN1
Cyclopropane SCHEMBL29022116 0.94 CYP1A2 (0.68) CYP1A2KDM4EHPGDCYP2C19MEN1
Dimethylformamide SCHEMBL11044579 0.86 CYP1A2 (0.58) CYP1A2KDM4EHPGDCYP2C19MEN1
SCHEMBL2068768 0.85 LMNA (0.68) CYP1A2KDM4EHPGDMEN1KMT2A
SCHEMBL29840068 0.85 GAA (0.67) CYP1A2KDM4EHPGDMEN1KMT2A
SCHEMBL3928666 0.85 GAA (0.67) CYP1A2KDM4EHPGDMEN1KMT2A
SCHEMBL6859262 0.84 CYP1A2 (0.64) CYP1A2KDM4EHPGDCYP2C19MEN1
SCHEMBL10458447 0.84 KDM4E (0.72) CYP1A2KDM4EHPGDCYP2C19MEN1
SCHEMBL4359338 0.84 CYP1A2 (0.56) CYP1A2KDM4EHPGDCYP2C19MEN1
SCHEMBL4107106 0.83 CYP1A2 (0.70) CYP1A2KDM4EHPGDCYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 203 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9198426-B2 Use of 5 pyridin-4-yl-1,3-thiazoles for controlling phytopathogenic fungi BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-12-01 US claimed
EP-2836485-A1 CONFORMATIONALLY CONSTRAINED, FULLY SYNTHETIC MACROCYCLIC COMPOUNDS Polyphor Ag (CH) 2015-02-18 EP claimed
WO-2013139697-A1 CONFORMATIONALLY CONSTRAINED, FULLY SYNTHETIC MACROCYCLIC COMPOUNDS POLYPHOR AG (CH) 2013-09-26 WO claimed
US-20100168185-A1 Use of 5-pyridin-4-yl-1,3-thiazoles for controlling phytopathogenic fungi BAYER CORPSCIENCE AG (DE) 2010-07-01 US claimed
EP-2198710-A1 Use of 5-pyridin-4yl-(1,3) thiazoles for combating phytopathogenic fungi Bayer CropScience AG (DE) 2010-06-23 EP claimed
CN-100389104-C Process for preparation of 2,6-dichloroaniline UNIV ZHEJIANG (CN) 2008-05-21 CN claimed
CN-1942475-A Substituted thieno - and thiazolo - [2, 3-d] pyridines as inhibitors of Tie2 ASTRAZENECA AB (SE) 2007-04-04 CN claimed
EP-1737830-A1 TRI-SUBSTITUTED UREAS AS CYTOKINE INHIBITORS The Procter and Gamble Company (US) 2007-01-03 EP claimed
EP-1716155-A1 SUBSTITUTED THIENO¬2,3-D|PYRIMIDINES AS INHIBITORS OF TIE2 AstraZeneca AB (SE) 2006-11-02 EP claimed
CN-1827584-A Process for preparation of 2,6-dichloroaniline UNIV ZHEJIANG (CN) 2006-09-06 CN claimed
WO-2005105757-A1 TRI-SUBSTITUTED UREAS AS CYTOKINE INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2005-11-10 WO claimed
EP-1578751-A1 PYRROLOPYRIMIDINE DERIVATIVES Pfizer Products Inc. (US) 2005-09-28 EP claimed
WO-2005075483-A1 SUBSTITUTED THIENO - AND THIAZOLO - [2, 3-D] PYRIDINES AS INHIBITORS OF TIE2 ASTRAZENECA AB (SE) 2005-08-18 WO claimed
WO-2004056830-A1 PYRROLOPYRIMIDINE DERIVATIVES PFIZER PRODUCTS INC. (US) 2004-07-08 WO claimed
JP-62018460-A None JP disclosed
US-12378354-B2 Active ester resin, method for producing thereof, epoxy resin composition, cured product thereof, prepreg, laminated board, and material for circuit substrate NIPPON STEEL CHEMICAL & MATERIAL CO., LTD. (JP) 2025-08-05 US disclosed
CN-119948080-A Active ester resin, epoxy resin composition, cured product thereof, prepreg, laminated board and laminated film 日铁化学材料株式会社 2025-05-06 CN disclosed
CN-85108862-A The preparation method and the application thereof of N-(3-chloro-1,2,4- diazole-5-yl) urea 1986-07-30 CN disclosed
EP-0182166-A2 Process for preparing phenylisopropylurea compounds AMERICAN CYANAMID COMPANY (US) 1986-05-28 EP disclosed
US-4578513-A Process for preparing phenylisopropylurea compounds AMERICAN CYANAMID COMPANY (US) 1986-03-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168185-A1 Use of 5-pyridin-4-yl-1,3-thiazoles for controlling phytopathogenic fungi PIR, PNPO, PDXK CYP1A2 1420/4885KDM4E 941/4885HPGD 2948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.