SCHEMBL21765829

SCHEMBL21765829

CC(C)(C=O)n1cccc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PCSK9 Q8NBP7 1/20 0.40
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
CHEK1 O14757 1/20 0.35
MAP4K4 O95819 1/20 0.35
CSF1R P07333 1/20 0.35
PRKACA P17612 1/20 0.35
KDR P35968 1/20 0.35
CDK8 P49336 1/20 0.35
MAP2K1 Q02750 1/20 0.35
ACVR1 Q04771 1/20 0.35
MAP4K2 Q12851 1/20 0.35
ROCK1 Q13464 1/20 0.35
DYRK1A Q13627 1/20 0.35
AURKB Q96GD4 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
TSHR P16473 1/20 0.35
ALDH1A1 P00352 5/20 0.33
MAPT P10636 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21747386 0.76 MEN1 (0.44) PCSK9KMT2AMEN1NPSR1ALDH1A1
SCHEMBL21747345 0.73 KMT2A (0.39) PCSK9KMT2AMEN1NPSR1ALDH1A1
SCHEMBL25544035 0.71 MEN1 (0.40) PCSK9KMT2AMEN1NPSR1TSHR
SCHEMBL27412445 0.71 PCSK9 (0.41) PCSK9KMT2AMEN1NPSR1CHEK1
Biphenyl SCHEMBL27538626 0.69 ALDH1A1 (0.47) ALDH1A1MAPTLMNAHTTCYP2C9
SCHEMBL21765754 0.69 KMT2A (0.45) KMT2AMEN1NPSR1ALDH1A1KDM4E
SCHEMBL6445284 0.67 PCSK9 (0.41) PCSK9CHEK1MAP4K4CSF1RPRKACA
SCHEMBL6444709 0.63 PCSK9 (0.73) PCSK9KMT2ANPSR1CHEK1MAP4K4
Formamide SCHEMBL28739639 0.62 ATM (0.52) PCSK9KMT2AMEN1ALDH1A1MAPT
SCHEMBL8634800 0.62 PCSK9 (0.44) PCSK9ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3613742-A1 INDOLIZINE DERIVATIVES AND APPLICATION THEREOF IN MEDICINE Kind Pharmaceutical (CN) 2020-02-26 EP disclosed