SCHEMBL27412445

SCHEMBL27412445

FC(F)(F)n1cccc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PCSK9 Q8NBP7 1/20 0.41
PTGS1 P23219 1/20 0.37
KIF11 P52732 1/20 0.37
KDR P35968 3/20 0.36
MAP4K4 O95819 2/20 0.36
PRKACA P17612 2/20 0.36
CDK8 P49336 2/20 0.36
MAP2K1 Q02750 2/20 0.36
MAP4K2 Q12851 2/20 0.36
ROCK1 Q13464 2/20 0.36
DYRK1A Q13627 2/20 0.36
AURKB Q96GD4 2/20 0.36
DYRK1B Q9Y463 2/20 0.36
CHEK1 O14757 1/20 0.36
CSF1R P07333 1/20 0.36
ACVR1 Q04771 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
XBP1 P17861 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27463283 0.75 PTGS2 (0.55) PTGS1KIF11
SCHEMBL21747386 0.72 MEN1 (0.44) PCSK9KDM4EMAPTXBP1MAPK1
SCHEMBL21765829 0.71 PCSK9 (0.40) PCSK9KDRMAP4K4PRKACACDK8
SCHEMBL28009342 0.71 GABRA1 (0.46) PTGS1KDM4EMAPTMAPK1ALDH1A1
SCHEMBL28277444 0.70 PCSK9 (0.45) PCSK9PTGS1KDRMAP4K4PRKACA
SCHEMBL21747345 0.66 KMT2A (0.39) PCSK9KIF11KDM4EMAPTALDH1A1
SCHEMBL11623898 0.65 ESR1 (0.42) KDRMAP4K4PRKACACDK8MAP2K1
SCHEMBL8881198 0.65 PCSK9 (0.45) PCSK9KDRMAP4K4PRKACACDK8
SCHEMBL9019096 0.65 PCSK9 (0.45) PCSK9PTGS1KDRMAP4K4PRKACA
SCHEMBL16152323 0.65 PCSK9 (0.45) PCSK9KDRMAP4K4PRKACACDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1074439-A A kind of method from the synthetic trifluoromethyl pyrpole compounds of trifluoromethyl  oxazolone SHANGHAI INST ORGANIC CHEM (CN) 1993-07-21 CN disclosed