SCHEMBL21766079

SCHEMBL21766079

COc1ccccc1CNC(=O)C1CCN(S(=O)(=O)c2cc(C)cc(C)c2)CC1

nearest known ligand 0.72

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.72
CYP2C19 P33261 2/20 0.72
CYP1A2 P05177 1/20 0.72
TSHR P16473 1/20 0.72
HPGD P15428 1/20 0.71
LMNA P02545 2/20 0.69
PKM P14618 2/20 0.69
TP53 P04637 1/20 0.68
POLB P06746 1/20 0.68
MAPT P10636 1/20 0.66
KMT2A Q03164 3/20 0.65
USP2 O75604 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
CYP3A4 P08684 1/20 0.64
PLA2G1B P04054 1/20 0.64
ATG4B Q9Y4P1 1/20 0.64
EPHX2 P34913 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20258825 0.89 ALDH1A1 (0.71) ALDH1A1CYP2C19CYP1A2TSHRHPGD
SCHEMBL20258782 0.89 ALDH1A1 (0.71) ALDH1A1CYP2C19CYP1A2TSHRHPGD
SCHEMBL21766087 0.86 PKM (0.78) PKMTP53KMT2APLA2G1BATG4B
SCHEMBL21765928 0.79 TP53 (0.82) ALDH1A1CYP2C19LMNAPKMTP53
SCHEMBL21765932 0.79 GAA (0.53) CYP2C19TSHRLMNAPKMPOLB
SCHEMBL5243818 0.79 MEN1 (0.67) ALDH1A1LMNAPKMTP53POLB
SCHEMBL21800686 0.78 ALDH1A1 (0.71) ALDH1A1CYP2C19CYP1A2TSHRHPGD
SCHEMBL20258778 0.78 PKM (0.69) ALDH1A1LMNAPKMTP53PLA2G1B
SCHEMBL21800651 0.77 ALDH1A1 (0.71) ALDH1A1CYP2C19CYP1A2TSHRHPGD
SCHEMBL21765931 0.77 SLC13A5 (0.82) ALDH1A1TP53POLBMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10793522-B2 Sulfonamides as inhibitors of the uptake of extracellular citrate BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-10-06 US disclosed
US-20200062708-A1 SULFONAMIDES AS INHIBITORS OF THE UPTAKE OF EXTRACELLULAR CITRATE BOEHRINGER INGELHEIM PHARMA GBMH & CO KG (DE) 2020-02-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200062708-A1 SULFONAMIDES AS INHIBITORS OF THE UPTAKE OF EXTRACELLULAR CITRATE CS, GLS, GLS2 ALDH1A1 732/4885CYP2C19 978/4885CYP1A2 843/4885
US-10793522-B2 Sulfonamides as inhibitors of the uptake of extracellular citrate CS, GLS, GLS2 ALDH1A1 732/4885CYP2C19 978/4885CYP1A2 843/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.