SCHEMBL21769359

SCHEMBL21769359

Cc1ccc(S(=O)ONC(=O)OC(C)(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.43
TDP1 Q9NUW8 2/20 0.38
MAPT P10636 3/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
RAB9A P51151 2/20 0.35
MIF P14174 1/20 0.34
TP53 P04637 1/20 0.34
GRM6 O15303 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23616359 0.78 NFKB1 (0.40) MAPTCA12CA1CA2CA9
SCHEMBL12067919 0.75 TDP1 (0.52) TDP1MAPTPPARGPPARACA12
SCHEMBL21161629 0.73 CA12 (0.49) RECQLTDP1MAPTCA12CA1
SCHEMBL21161191 0.73 CA12 (0.49) RECQLTDP1MAPTCA12CA1
SCHEMBL21161661 0.73 CA12 (0.49) RECQLTDP1MAPTCA12CA1
SCHEMBL23966869 0.72 RECQL (0.38) RECQLTDP1PPARGPPARACYP1A2
SCHEMBL19675061 0.71 ALDH1A1 (0.42) RECQLTDP1MAPTRAB9ACYP1A2
SCHEMBL29167216 0.71 ALDH1A1 (0.42) RECQLTDP1MAPTRAB9ACYP1A2
SCHEMBL17147606 0.71 PPARG (0.39) TDP1MAPTPPARGPPARACA12
SCHEMBL178373 0.70 CYP17A1 (0.54) TDP1MAPTCA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3197276-B1 HERBICIDAL PYRIDINO-/PYRIMIDINO-THIAZOLES SYNGENTA PARTICIPATIONS AG (CH) 2023-06-07 EP disclosed
EP-3772516-B1 TROPOMYOSIN RECEPTOR KINASE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF JIANGSU VCARE PHARMATECH CO LTD (CN) 2022-12-14 EP disclosed
EP-3842425-A1 NOVEL QUINOLINE DERIVATIVE INHIBITOR Nanjing Transthera Biosciences Co., Ltd. (CN) 2021-06-30 EP disclosed
EP-3772516-A1 TROPOMYOSIN RECEPTOR KINASE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF Jiangsu Vcare Pharmatech Co., Ltd (CN) 2021-02-10 EP disclosed
WO-2020038460-A1 NOVEL QUINOLINE DERIVATIVE INHIBITOR 南京药捷安康生物科技有限公司 2020-02-27 WO disclosed