SCHEMBL23616359

SCHEMBL23616359

Cc1cc(C)c(S(=O)ONC(=O)OC(C)(C)C)c(C)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
LCK P06239 7/20 0.39
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA9 Q16790 2/20 0.34
CA2 P00918 1/20 0.34
NLRP3 Q96P20 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CISD2 Q8N5K1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21769359 0.78 RECQL (0.43) CYP2C19ALDH1A1MAPTTSHRCA12
SCHEMBL22959260 0.71 RAPGEF4 (0.34) ALDH1A1CA1CA2NLRP3SMN1; SMN2
SCHEMBL25822650 0.71 NFKB1 (0.40) NFKB1NFKB2RELALCKCYP2C9
SCHEMBL3131919 0.70 LCK (0.60) NFKB1NFKB2RELALCKALDH1A1
SCHEMBL25047 0.70 NFKB1 (0.42) NFKB1NFKB2RELALCKMAPT
Glycine SCHEMBL27580905 0.69 LMNA (0.54) NFKB1NFKB2RELALCKALDH1A1
SCHEMBL22666755 0.67 CA1 (0.33) ALDH1A1MAPTCA1CA2NLRP3
SCHEMBL11181297 0.67 KDM4E (0.32) ALDH1A1MAPTTSHR
SCHEMBL31636878 0.67 NFKB1 (0.40) NFKB1NFKB2RELALCKNPSR1
SCHEMBL23453153 0.66 CA12 (0.50) LCKMAPTCA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4201936-A1 HETEROAROMATIC RING COMPOUND AS RET KINASE INHIBITOR, AND PREPARATION AND USE THEREOF Jiangsu Chia Tai Fenghai Pharmaceutical Co., Ltd. (CN) 2023-06-28 EP disclosed
EP-3992197-A1 NITROGEN-CONTAINING POLYCYCLIC FUSED RING COMPOUNDS, AND PHARMACEUTICAL COMPOSITION THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Applied Pharmaceutical Science, Inc. (CN) 2022-05-04 EP disclosed
EP-3845531-A1 SUBSTITUTED PYRAZOLE FUSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF Applied Pharmaceutical Science, Inc. (CN) 2021-07-07 EP disclosed