Phthalimide

Phthalimide

SCHEMBL217772

CS(=O)(=O)O.O=C1NC(=O)c2ccccc21

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of Phthalimide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB known ✓ P27338 1/20 0.45
EGFR known ✓ P00533 1/20 0.42
GSK3B P49841 1/20 0.68
CASP3 P42574 4/20 0.64
CASP2 P42575 1/20 0.64
CASP7 P55210 1/20 0.64
CASP6 P55212 1/20 0.64
CASP8 Q14790 1/20 0.64
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
ALDH1A1 P00352 4/20 0.47
HPGD P15428 4/20 0.47
LMNA P02545 4/20 0.47
MAPT P10636 3/20 0.47
BLM P54132 3/20 0.47
APAF1 O14727 1/20 0.47
THRB P10828 1/20 0.47
PARP1 P09874 2/20 0.45
MAOA P21397 1/20 0.45
PDGFRA P16234 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phthalimide SCHEMBL7164645 1.00 GSK3B (0.68) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL29217853 0.91 GSK3B (0.75) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL27968411 0.91 GSK3B (0.75) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL28035222 0.86 GSK3B (0.68) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL28035221 0.86 GSK3B (0.68) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL3220884 0.86 GSK3B (0.68) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL23063638 0.83 GSK3B (0.88) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL64 0.83 GSK3B (1.00) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL29366030 0.83 GSK3B (1.00) GSK3BCASP3CASP2CASP7CASP6
Phthalimide SCHEMBL11040503 0.83 GSK3B (1.00) GSK3BCASP3CASP2CASP7CASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096478-A Resist material for forming a chemically amplified negative type resist pattern and method of manufacturing a semiconductor device employing the resist pattern NEC CORPORATION (JP) 2000-08-01 US claimed
CN-107924131-A Material for forming underlayer film for lithography, composition for forming underlayer film for lithography, method for producing same, and method for forming resist pattern 三菱瓦斯化学株式会社 2018-04-17 CN disclosed
CN-107533297-A Material for forming underlayer film for lithography, composition for forming underlayer film for lithography, and pattern formation method 三菱瓦斯化学株式会社 2018-01-02 CN disclosed
CN-107430344-A Lower layer film for lithography, which forms to be formed with material, lower layer film for lithography, uses composition, lower layer film for lithography and pattern formation method 三菱瓦斯化学株式会社 2017-12-01 CN disclosed
CN-106575083-A Underlayer film-forming composition for lithography, underlayer film for lithography, and pattern forming method 三菱瓦斯化学株式会社 2017-04-19 CN disclosed
CN-106103396-A Compound, resin, lower layer film for lithography form material, lower layer film for lithography, pattern formation method and compound or the purification process of resin 三菱瓦斯化学株式会社 2016-11-09 CN disclosed
EP-1788436-B1 Rework process for photoresist film SHINETSU CHEMICAL CO (JP) 2013-01-09 EP disclosed
EP-1813985-B1 Antireflection film composition, substrate, and pattering process SHINETSU CHEMICAL CO (JP) 2012-10-31 EP disclosed
US-8288072-B2 Antireflection film; fast etching speed whcih reduces deformation; accuracy; 2,3-epoxypropyl methacrylate ester-styrene copolymer SHIN-ETSU CHEMICAL CO., LTD. (JP) 2012-10-16 US disclosed
US-8088554-B2 Bottom resist layer composition and patterning process using the same SHIN-ETSU CHEMICAL CO., LTD (JP) 2012-01-03 US disclosed
US-20050079446-A1 Novel polymerizable compound, polymer, positive-resist composition, and patterning process using the same SHIN-ETSU CHEMICAL CO., LTD. (JP) 2005-04-14 US disclosed
US-20050014092-A1 Novel compound, polymer, resist composition, and patterning process SHIN-ETSU CHEMICAL CO., LTD. (JP) 2005-01-20 US disclosed
US-20040259037-A1 Resist lower layer film material and method for forming a pattern SHIN-ETSU CHEMICAL CO., LTD. (JP) 2004-12-23 US disclosed
US-20040241577-A1 Resist lower layer film material and method for forming a pattern SHIN-ETSU CHEMICAL CO., LTD. (JP) 2004-12-02 US disclosed
EP-1482361-A1 ACID-DEGRADABLE RESIN COMPOSITIONS CONTAINING KETENE-ALDEHYDE COPOLYMER NIPPON SODA CO., LTD. (JP) 2004-12-01 EP disclosed
US-20020028943-A1 Multibinding inhibitors of microsomal triglyceride transferase protein THERAVANCE BIOPHARMA R&D IP, LLC 2002-03-07 US disclosed
US-6288234-B1 FLUORINATED HETEROCYCLIC AMIDO AMINE COMPOUNDS AS DRUGS ADVANCED MEDICINE, INC. 2001-09-11 US disclosed
EP-1085846-A2 MULTIBINDING INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFERASE PROTEIN Advanced Medicine, Inc. (US) 2001-03-28 EP disclosed
WO-1999063929-A9 MULTIBINDING INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFERASE PROTEIN ADVANCED MEDICINE INC (US) 2000-03-16 WO disclosed
WO-1999063929-A2 MULTIBINDING INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFERASE PROTEIN ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020028943-A1 Multibinding inhibitors of microsomal triglyceride transferase protein MTTP, CETP, HDLBP MAOB 1607/4885EGFR 4755/4885GSK3B 3060/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.