SCHEMBL21779370

SCHEMBL21779370

Fc1cc(F)c(COC2CCCC2)cc1F

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.45
SCN9A Q15858 3/20 0.44
HTR2C P28335 2/20 0.40
SLC6A4 P31645 2/20 0.40
HTR2A P28223 1/20 0.40
HTR1A P08908 1/20 0.39
NAAA Q02083 7/20 0.38
KDM4E B2RXH2 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CARM1 Q86X55 1/20 0.35
PRMT6 Q96LA8 1/20 0.35
DRD4 P21917 2/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3126431 0.84 HTR1A (0.37) DPP4SCN9AHTR2CSLC6A4HTR2A
SCHEMBL22283641 0.79 NAAA (0.40) DPP4SCN9AHTR1ANAAA
SCHEMBL22283644 0.79 NAAA (0.40) DPP4SCN9AHTR1ANAAA
SCHEMBL28391073 0.78 NAAA (0.40) DPP4HTR1ANAAA
SCHEMBL18615735 0.78 NAAA (0.59) SCN9AHTR1ANAAAKDM4EL3MBTL1
SCHEMBL30198976 0.76 CXCR3 (0.49) SCN9ANAAAKDM4EL3MBTL1DRD4
SCHEMBL18615766 0.76 CARM1 (0.57) HTR2CSLC6A4HTR2AHTR1AKDM4E
SCHEMBL15536664 0.74 SCN9A (0.54) DPP4SCN9AHTR1ANAAAKDM4E
SCHEMBL2101438 0.74 NAAA (0.59) HTR1ANAAAKDM4EL3MBTL1CARM1
SCHEMBL18579558 0.74 DPP4 (0.40) DPP4HTR2CSLC6A4HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3344613-B1 HETEROARYL COMPOUNDS AND THEIR USE AS THERAPEUTIC DRUGS DONG A SOCIO HOLDINGS CO LTD (KR) 2020-03-04 EP disclosed