SCHEMBL21780155

SCHEMBL21780155

CC1COC2Cn3ccc(=O)c(OCc4ccccc4)c3C(=O)N12

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 2/20 0.42
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 2/20 0.42
HPGD P15428 1/20 0.42
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 1/20 0.37
GRM2 Q14416 1/20 0.36
GLRA1 P23415 1/20 0.32
S1PR5 Q9H228 1/20 0.32
NAAA Q02083 1/20 0.31
HTR2C P28335 1/20 0.31
MAPK14 Q16539 1/20 0.31
PDE4B Q07343 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2160801 1.00 HTT (0.42) HTTSMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL2298978 0.90 HTT (0.41) HTTSMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL2161654 0.82 GRM2 (0.36) HTTSMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL21780072 0.82 GRM2 (0.36) HTTSMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL12239929 0.82 HTT (0.43) HTTSMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL24969604 0.81 SLC22A2 (0.39) LMNAGRM2GLRA1S1PR5
SCHEMBL21780077 0.79 ALDH1A1 (0.41) HTTSMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL24969606 0.79 SLC22A2 (0.41) HTTMEN1ALDH1A1KMT2AHPGD
SCHEMBL21780078 0.78 HTT (0.40) HTTSMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL12239939 0.78 HTT (0.39) HTTSMN1; SMN2MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617194-A1 PROCESSES AND INTERMEDIATES FOR CARBAMOYLPYRIDONE HIV INTEGRASE INHIBITORS VIIV Healthcare Company (US) 2020-03-04 EP disclosed