SCHEMBL21780327

SCHEMBL21780327

CCC(CO)(CBr)NC(C)=O

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.40
KDM4E B2RXH2 1/20 0.40
THRB P10828 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18622068 0.87 PKM (0.45) PKMKDM4ETHRBHRH3HTT
SCHEMBL9816463 0.79 KDM4E (0.45) PKMKDM4ETHRBHRH3HTT
SCHEMBL14366070 0.79 KDM4E (0.40) PKMKDM4ETHRBHTT
SCHEMBL20388578 0.79 PKM (0.40) PKMKDM4ETHRBHRH3HTT
SCHEMBL14885080 0.71 PKM (0.38) PKMKDM4ETHRBHTT
SCHEMBL8853319 0.71 L3MBTL1 (0.32)
SCHEMBL25763081 0.70 HRH3 (0.35) PKMKDM4EHRH3
SCHEMBL4578255 0.69 KDM4E (0.36) PKMKDM4EHRH3
SCHEMBL15972133 0.69 KDM4E (0.36) PKMKDM4EHRH3
SCHEMBL14136486 0.68 PKM (0.41) PKMKDM4ETHRBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3097098-B1 PROCESS FOR THE PREPARATION OF N-[(3-AMINOOXETAN-3-YL)METHYL]-2-(1,1-DIOXO-3,5-DIHYDRO-1,4-BENZOTHIAZEPIN-4-YL)-6-METHYL-QUINAZOLIN-4-AMINE HOFFMANN LA ROCHE (CH) 2020-03-04 EP disclosed