SCHEMBL21780491

SCHEMBL21780491

COC1=CCC=C(c2ccc(C(C)(C)F)cc2)C=C1C(=O)N1CCN(Cc2ncccn2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 4/20 0.37
SLC6A7 Q99884 2/20 0.37
MAPT P10636 2/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
LSS P48449 1/20 0.36
STAT3 P40763 2/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
SIGMAR1 Q99720 1/20 0.36
PRKAA2 P54646 2/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21780429 0.76 KCNK3 (0.46) KDM4EALDH1A1PTGDR2MEN1KMT2A
SCHEMBL21780486 0.69 PTGDR2 (0.47) KDM4EALDH1A1SLC6A7TSHRPTGDR2
SCHEMBL21780432 0.60 TLR9 (0.43) KDM4EALDH1A1TSHRKMT2AKCNK3
SCHEMBL17886713 0.59 ALDH1A1 (0.72) KDM4EALDH1A1MAPTTSHRMAPK1
SCHEMBL21780503 0.59 KCNK3 (0.43) ALDH1A1TSHRKCNK3KCNK9PIK3CA
SCHEMBL15853631 0.57 RORC (0.64) KDM4EALDH1A1MAPTTSHRMAPK1
SCHEMBL15853648 0.56 RORC (0.65) KDM4EALDH1A1KMT2AKCNK3KCNK9
SCHEMBL15853630 0.56 RORC (0.62) LSSSIGMAR1
SCHEMBL21780426 0.55 KMT2A (0.53) ALDH1A1TSHRMEN1KMT2AHTT
SCHEMBL13974784 0.55 RORC (0.65) KDM4EALDH1A1LSSMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3085696-B1 FUSED BENZOXAZEPINONES AS ION CHANNEL MODULATORS GILEAD SCIENCES INC (US) 2020-03-04 EP disclosed