SCHEMBL21780744

SCHEMBL21780744

CCc1ccc(OC)cc1C#N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
GLA P06280 2/20 0.46
HSD17B10 Q99714 4/20 0.46
TP53 P04637 2/20 0.46
KDM4E B2RXH2 5/20 0.46
MAPT P10636 5/20 0.46
L3MBTL1 Q9Y468 4/20 0.46
ALDH1A1 P00352 4/20 0.46
CASP1 P29466 2/20 0.46
CLK1 P49759 2/20 0.46
MAPK1 P28482 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
CASP7 P55210 1/20 0.46
NPY1R P25929 1/20 0.46
NPY2R P49146 1/20 0.46
MAOB P27338 1/20 0.43
GAA P10253 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7672592 0.87 NPC1 (0.46) NPC1RAB9AMEN1KMT2AGLA
SCHEMBL7672598 0.85 NPC1 (0.47) NPC1RAB9AMEN1KMT2AGLA
SCHEMBL13652097 0.85 NOS2 (0.51) NPC1RAB9AMEN1KMT2AGLA
SCHEMBL1488919 0.84 NPC1 (0.43) NPC1RAB9AMEN1KMT2AGLA
SCHEMBL2085379 0.84 NPC1 (0.43) NPC1RAB9AMEN1KMT2AGLA
SCHEMBL2441387 0.82 HSD17B10 (0.58) NPC1RAB9AMEN1KMT2AGLA
SCHEMBL16959547 0.81 APLNR (0.41) HSD17B10MAPTL3MBTL1ALDH1A1POLB
SCHEMBL21728056 0.81 LMNA (0.43) NPC1RAB9AMEN1KMT2AGLA
SCHEMBL27279821 0.81 NPC1 (0.41) NPC1RAB9AMEN1KMT2AGLA
SCHEMBL2437800 0.80 NPC1 (0.55) NPC1RAB9AMEN1KMT2AGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3402781-B1 3-((HETERO-)ARYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES GRUENENTHAL GMBH (DE) 2020-03-04 EP disclosed