SCHEMBL21780801

SCHEMBL21780801

CCCN(CCC)C(=O)c1ncc(C)cn1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.47
LPAR1 Q92633 1/20 0.40
LPAR5 Q9H1C0 1/20 0.40
MLYCD O95822 1/20 0.40
SPR P35270 2/20 0.39
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38
POLB P06746 1/20 0.38
APEX1 P27695 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
CA12 O43570 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
APLNR P35414 1/20 0.36
HCAR3 P49019 2/20 0.36
CRHR1 P34998 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15780518 0.74 APLNR (0.41) SPRALDH1A1HPGDAPLNR
SCHEMBL19144976 0.73 OPRM1 (0.41) POLBAPLNR
SCHEMBL10783583 0.71 TP53 (0.44) TP53LPAR1LPAR5MLYCDSPR
SCHEMBL30778096 0.71 TP53 (0.37) TP53LPAR1LPAR5MLYCDSPR
SCHEMBL5429491 0.70 MLYCD (0.51) TP53MLYCDEGFRERBB2HPGD
SCHEMBL15148333 0.70 APLNR (0.41) TDP1ALDH1A1APLNR
SCHEMBL14141210 0.69 TP53 (0.50) TP53MLYCDEGFRERBB2TDP1
SCHEMBL7967022 0.69 MLYCD (0.64) TP53MLYCDEGFRERBB2ALDH1A1
SCHEMBL17580501 0.69 EGFR (0.42) TP53EGFRERBB2ALDH1A1HPGD
SCHEMBL19550744 0.68 APLNR (0.37) MLYCDTDP1ALDH1A1APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3402781-B1 3-((HETERO-)ARYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES GRUENENTHAL GMBH (DE) 2020-03-04 EP disclosed