SCHEMBL21780873

SCHEMBL21780873

O=C(OCc1ccccc1)c1c(-c2ccccc2)sc2cc(O)ccc12

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.51
ESR2 Q92731 7/20 0.51
AKR1B1 P15121 1/20 0.47
LMNA P02545 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
HDAC3 O15379 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC8 Q9BY41 2/20 0.45
NCOR2 Q9Y618 2/20 0.45
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21780715 0.90 LMNA (0.47) ESR1ESR2AKR1B1LMNANPC1
SCHEMBL21780868 0.87 TDP1 (0.53) ESR1ESR2LMNANPC1SLC6A2
SCHEMBL11547729 0.80 ESR1 (0.68) ESR1ESR2KMT2ATDP1
SCHEMBL7107598 0.76 ESR1 (0.75) ESR1ESR2KMT2ATDP1
SCHEMBL5456037 0.74 MAOA (0.45) ESR1ESR2AKR1B1NPC1RAB9A
SCHEMBL11546633 0.74 ESR1 (0.67) ESR1ESR2LMNASLC6A2SLC6A3
SCHEMBL30898314 0.72 ESR1 (0.65) ESR1ESR2LMNAHDAC1SLC6A2
SCHEMBL11550840 0.72 CNR1 (0.71) ESR1ESR2LMNASLC6A2SLC6A3
SCHEMBL21940625 0.70 KMT2A (0.50) LMNANPC1RAB9ASLC6A2SLC6A3
SCHEMBL11551107 0.69 CNR1 (0.67) ESR1ESR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233828-B1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2020-03-04 EP disclosed