SCHEMBL21782008

SCHEMBL21782008

CCCC(=O)NCC(=O)NC(CCCNC(N)=O)C(=O)Nc1ccc(CCNC=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.44
CHRNB4 P30926 2/20 0.44
CHRNA3 P32297 2/20 0.44
CHRNA4 P43681 2/20 0.44
SIRT1 Q96EB6 2/20 0.40
GRIA1 P42261 7/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
CHRNA1 P02708 1/20 0.39
CHRNG P07510 1/20 0.39
CHRNB1 P11230 1/20 0.39
GRIN1 Q05586 1/20 0.39
CHRND Q07001 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRM1 Q13255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21649652 0.88 SIRT1 (0.42) CHRNB2CHRNB4CHRNA3CHRNA4SIRT1
SCHEMBL22593891 0.85 TRPV1 (0.45) GRIA1CHRNA1CHRNGCHRNB1CHRND
SCHEMBL21782007 0.84 C3AR1 (0.37) SIRT1SIRT2
SCHEMBL21782108 0.82 SPHK1 (0.37)
SCHEMBL23838548 0.81 SIRT1 (0.37) SIRT1GRIA1SIRT2
SCHEMBL22593908 0.81 TRPV1 (0.46) SIRT1GRIA1SIRT2
SCHEMBL22561449 0.81 C3AR1 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4SIRT1
SCHEMBL22214485 0.80 SIRT2 (0.46) SIRT1GRIA1SIRT2
SCHEMBL22593910 0.79 TRPV1 (0.46)
SCHEMBL25765429 0.77 NPY5R (0.40) SIRT1SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed