SCHEMBL22561449

SCHEMBL22561449

CCOCC(=O)NCC(=O)NC(CCCNC(N)=O)C(=O)Nc1ccc(CNC=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 1/20 0.43
HPGD P15428 2/20 0.38
ALDH1A1 P00352 1/20 0.38
SIRT2 Q8IXJ6 8/20 0.38
SIRT1 Q96EB6 8/20 0.38
FURIN P09958 2/20 0.36
NAMPT P43490 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
SIRT3 Q9NTG7 3/20 0.34
NPY1R P25929 1/20 0.34
ADAM10 O14672 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP12 P39900 1/20 0.34
MMP14 P50281 1/20 0.34
ADAM8 P78325 1/20 0.34
ADAM17 P78536 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21782007 0.86 C3AR1 (0.37) C3AR1SIRT2SIRT1NPY1RADAM10
SCHEMBL21781914 0.81 SPHK1 (0.42) C3AR1SIRT1NPY1RADAM10MMP2
SCHEMBL21782008 0.81 CHRNB2 (0.44) SIRT2SIRT1CHRNB2CHRNB4CHRNA3
SCHEMBL21649652 0.77 SIRT1 (0.42) SIRT2SIRT1FURINCHRNB2CHRNB4
SCHEMBL26273239 0.76 SIRT2 (0.44) SIRT2SIRT1SIRT3
SCHEMBL25774207 0.76 SIRT2 (0.46) SIRT2SIRT1SIRT3
SCHEMBL22214485 0.75 SIRT2 (0.46) SIRT2SIRT1SIRT3
SCHEMBL22810892 0.75 SIRT2 (0.41) C3AR1SIRT2SIRT1SIRT3ADAM10
SCHEMBL22593891 0.75 TRPV1 (0.45) NPY1R
SCHEMBL18811657 0.74 CA1 (0.48) C3AR1SIRT2SIRT1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725798-A1 BIOACTIVE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-10-21 EP disclosed