SCHEMBL21782044

SCHEMBL21782044

CNC(Cc1ccccc1)C(=O)NCc1ccc(NC(=O)C(CCCN)NC(=O)CNC(=O)CCCN2CCC(C(N)=O)CC2C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP7 P09237 5/20 0.38
ITGB1 P05556 2/20 0.38
ITGA5 P08648 1/20 0.38
AKT1 P31749 3/20 0.38
HRH1 P35367 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
KDM1A O60341 1/20 0.36
ITGA4 P13612 1/20 0.36
ACE P12821 2/20 0.35
CALCRL Q16602 1/20 0.35
MMP2 P08253 1/20 0.35
MMP12 P39900 1/20 0.35
MMP14 P50281 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21782071 0.82 ITGB1 (0.34) MMP7ITGB1ITGA5AKT1KDM1A
SCHEMBL21781797 0.82 AKT1 (0.39) MMP7ITGB1ITGA5AKT1HRH1
SCHEMBL21782018 0.80 AKT1 (0.37) MMP7ITGB1ITGA5AKT1HRH1
SCHEMBL21781742 0.80 MMP7 (0.32) MMP7ITGB1ITGA5ITGA4
SCHEMBL21781814 0.75 AKT1 (0.31) ITGB1ITGA5AKT1
SCHEMBL21781807 0.73 CYP3A4 (0.31) ITGB1AKT1ITGA4
SCHEMBL21782047 0.73
SCHEMBL21781748 0.73 KMT2A (0.31) MMP7ITGB1ITGA5KMT2AMEN1
SCHEMBL21782101 0.71 AKT1 (0.39) ITGB1ITGA5AKT1KMT2AMEN1
SCHEMBL22068095 0.69 MAP1LC3B (0.36) ITGB1HRH1KMT2AMEN1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed