SCHEMBL21782835

SCHEMBL21782835

CCc1ccccc1NC(=O)c1c(N)cccc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.52
LMNA P02545 2/20 0.52
TP53 P04637 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
MAPT P10636 5/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ALDH1A1 P00352 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 2/20 0.48
KCNK3 O14649 1/20 0.48
KCNK9 Q9NPC2 1/20 0.48
HTT P42858 1/20 0.48
HDAC1 Q13547 2/20 0.46
GAA P10253 1/20 0.46
HDAC3 O15379 1/20 0.45
MAPK1 P28482 1/20 0.45
HDAC2 Q92769 1/20 0.45
RECQL P46063 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27635898 0.85 LMNA (0.55) PKMLMNATP53RXFP1MAPT
SCHEMBL10296668 0.83 HTT (0.63) LMNATP53ALDH1A1MEN1KMT2A
SCHEMBL25872127 0.81 MAPT (0.52) PKMLMNATP53RXFP1MAPT
SCHEMBL735325 0.80 CYP1A2 (0.51) PKMLMNATP53RXFP1MAPT
SCHEMBL29154642 0.78 KDM4E (0.60) LMNATP53RXFP1MAPTALDH1A1
SCHEMBL8424563 0.76 NPC1 (0.46) MEN1KMT2AHDAC1HPGD
SCHEMBL7183194 0.76 MAPT (0.55) LMNATP53RXFP1MAPTALDH1A1
SCHEMBL16346420 0.76 GAA (0.59) LMNAMAPTSMN1; SMN2ALDH1A1MEN1
SCHEMBL15014130 0.76 TAS1R3 (0.54) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL734053 0.74 TAS1R3 (0.59) LMNATP53MAPTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3029041-B1 INHIBITORS OF HUMAN PHOSPHATIDYL-INOSITOL 3-KINASE DELTA ICOS CORP (US) 2020-03-04 EP disclosed