SCHEMBL2179437

SCHEMBL2179437

CCCC(CCC)CN(C(=O)OC(C)(C)C)c1cccc(C(O)CCNC(=O)OC(C)(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.40
ITGA4 P13612 1/20 0.40
GPR88 Q9GZN0 2/20 0.37
NQO2 P16083 1/20 0.37
KCNA5 P22460 1/20 0.37
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA12 O43570 1/20 0.36
CA14 Q9ULX7 1/20 0.36
DRD2 P14416 2/20 0.35
BACE1 P56817 5/20 0.35
MALT1 Q9UDY8 1/20 0.34
CTSK P43235 2/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2821039 0.92 GPR88 (0.39) ITGB1ITGA4GPR88NQO2KCNA5
SCHEMBL2177713 0.83 BACE1 (0.44) ITGB1ITGA4BACE1CTSKMEN1
SCHEMBL2167444 0.81 EPHX1 (0.36) ITGB1ITGA4GPR88NQO2KCNA5
SCHEMBL2178099 0.79 IDO1 (0.42) ITGB1ITGA4BACE1CTSKMEN1
SCHEMBL1710754 0.77 GPR88 (0.39) GPR88NQO2KCNA5CA1CA2
SCHEMBL2176308 0.76 L3MBTL1 (0.50) BACE1
SCHEMBL2158118 0.76 SIGMAR1 (0.43) BACE1CTSK
SCHEMBL16031480 0.76 NQO2 (0.51) NQO2KCNA5CA1CA2MALT1
SCHEMBL16079975 0.76 POLB (0.45) GPR88NQO2KCNA5CA1CA2
SCHEMBL17735443 0.76 POLB (0.45) GPR88NQO2KCNA5CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340242-A2 COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2011-07-06 EP disclosed