SCHEMBL2179805

SCHEMBL2179805

COc1cnc2cc(C(Oc3ccc(Cl)cc3)c3ccc(S(C)(=O)=O)cc3)[nH]c2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.38
PTGS2 P35354 4/20 0.36
PTGS1 P23219 3/20 0.36
LRRK2 Q5S007 1/20 0.35
GCK P35557 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX15 P16050 1/20 0.35
NFKB1 P19838 1/20 0.35
HIF1A Q16665 1/20 0.35
GMNN O75496 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
APEX1 P27695 1/20 0.35
PMP22 Q01453 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2197573 0.91 PIK3CA (0.34) CNR2PTGS2PTGS1LRRK2GCK
SCHEMBL12490119 0.78 GCK (0.46) PTGS2PTGS1GCKALDH1A1POLB
SCHEMBL2178524 0.72 GCK (0.42) LRRK2GCK
SCHEMBL2178527 0.66 GCK (0.35) PTGS2PTGS1LRRK2GCKATR
SCHEMBL11568045 0.62 PTGS2 (0.44) CNR2PTGS2PTGS1GCKCYP11B1
SCHEMBL2197752 0.60 GCK (0.40) PTGS2PTGS1GCKMAPT
SCHEMBL7363201 0.59 PTGS2 (0.56) PTGS2PTGS1SMN1; SMN2CYP3A4ALDH1A1
SCHEMBL265232 0.59 PTGS2 (0.69) PTGS2PTGS1CYP3A4ALDH1A1
SCHEMBL31631767 0.59 PTGS2 (0.37) PTGS2PTGS1SMN1; SMN2TP53ALDH1A1
SCHEMBL940743 0.59 PTGS2 (0.57) PTGS2PTGS1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080755-A1 FUSED NITROGEN HETEROCYCLIC COMPOUNDS, PROCESS OF PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-07-07 WO claimed
WO-2011080755-A1 FUSED NITROGEN HETEROCYCLIC COMPOUNDS, PROCESS OF PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-07-07 WO disclosed