SCHEMBL2197573

SCHEMBL2197573

COc1cnc2cc(C(Oc3ccc(Cl)nc3)c3ccc(S(C)(=O)=O)cc3)[nH]c2n1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.34
GCK P35557 4/20 0.34
LRRK2 Q5S007 1/20 0.34
ATR Q13535 1/20 0.33
ALDH1A1 P00352 1/20 0.33
BLM P54132 1/20 0.33
PTGS2 P35354 5/20 0.32
PTGS1 P23219 2/20 0.32
EGFR P00533 1/20 0.32
PIK3CD O00329 1/20 0.31
PIK3CB P42338 1/20 0.31
PIK3CG P48736 1/20 0.31
CNR2 P34972 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2179805 0.91 CNR2 (0.38) PIK3CAGCKLRRK2ATRALDH1A1
SCHEMBL2178524 0.70 GCK (0.42) GCKLRRK2
SCHEMBL12490119 0.69 GCK (0.46) GCKALDH1A1PTGS2PTGS1
SCHEMBL2178905 0.66 GCK (0.38) GCK
SCHEMBL2178527 0.65 GCK (0.35) GCKLRRK2ATRPTGS2PTGS1
SCHEMBL1256644 0.60 SMN1; SMN2 (0.59) ALDH1A1BLMEGFR
SCHEMBL29977958 0.60 SMN1; SMN2 (0.59) ALDH1A1BLMEGFR
SCHEMBL6808653 0.59 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL4689890 0.58 SMN1; SMN2 (0.48) ALDH1A1
SCHEMBL602439 0.57 HCAR1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080755-A1 FUSED NITROGEN HETEROCYCLIC COMPOUNDS, PROCESS OF PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-07-07 WO claimed
WO-2011080755-A1 FUSED NITROGEN HETEROCYCLIC COMPOUNDS, PROCESS OF PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-07-07 WO disclosed