SCHEMBL2179938

SCHEMBL2179938

O=C=Nc1ccc2c(c1)C=CC2

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CYP3A4 P08684 2/20 0.41
TRPA1 O75762 1/20 0.41
TSHR P16473 1/20 0.37
CYP1A2 P05177 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14569468 0.79 CYP2D6 (0.31) MAPK1TDP1CYP3A4TSHRCYP1A2
SCHEMBL2497578 0.72 CA1 (0.33) CA1CA2
SCHEMBL275807 0.70 CA1 (0.33) CA1CA2
SCHEMBL11231604 0.69 MAPK1 (0.48) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL543138 0.69 MAPK1 (0.48) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL29561757 0.68 ALDH1A1 (0.38) TDP1TSHR
SCHEMBL30632049 0.68 ADRA2A (0.47) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL672098 0.68 ADRA2A (0.47) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL9629684 0.68 CA1 (0.34) CA1CA2
SCHEMBL15876269 0.67 CA1 (0.35) CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116829542-A Benzothiazole and benzimidazole derivatives, pharmaceutically acceptable salts, preparation method thereof and pharmaceutical composition containing same as active ingredient 韩国化学研究院 2023-09-29 CN disclosed
CN-107849816-B Method for treating paperboard and paper media and related treated paperboard and paper media 巴斯夫欧洲公司 2021-07-09 CN disclosed
EP-2519500-A1 INHIBITORS OF DIACYLGLYCEROL ACYL TRANSFERASE Piramal Healthcare Ltd. (IN) 2012-11-07 EP disclosed
WO-2011080718-A1 INHIBITORS OF DIACYLGLYCEROL ACYL TRANSFERASE PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-07-07 WO disclosed