SCHEMBL2180713

SCHEMBL2180713

Cc1cnc(O)c2nccn12

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.32
CCNE2 O96020 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
IKBKB O14920 1/20 0.31
KDM4E B2RXH2 2/20 0.30
MAPT P10636 2/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
HTT P42858 1/20 0.30
NUDT1 P36639 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20382914 0.92 TLR7 (0.33) KDM4EMAPTALDH1A1GAAHTT
SCHEMBL15918975 0.81 PDE10A (0.36) L3MBTL1IKBKBNUDT1
SCHEMBL21986320 0.78 L3MBTL1 (0.34) L3MBTL1IKBKB
SCHEMBL2480217 0.78 NUDT1 (0.47) NUDT1
SCHEMBL2180681 0.78 GRIN2D (0.33) CCNE2CCNE1CDK2L3MBTL1IKBKB
SCHEMBL14381040 0.77 TLR7 (0.33)
SCHEMBL19554107 0.76 MYC (0.38) SSTR4L3MBTL1KDM4EMAPTALDH1A1
SCHEMBL15061729 0.73 TLR7 (0.32)
SCHEMBL22337979 0.73 SSTR4 (0.39) SSTR4CCNE2CCNE1CDK2IKBKB
SCHEMBL8240025 0.73 TLR7 (0.53) NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2567960-A2 Imidazo[1,2-a]pyrazine compounds for treatment of viral infections such as hepatitis Biofocus DPI Limited (GB) 2013-03-13 EP disclosed
EP-2567960-A2 Imidazo[1,2-a]pyrazine compounds for treatment of viral infections such as hepatitis Biofocus DPI Limited (GB) 2013-03-13 EP disclosed
EP-2193131-B1 IMIDAZO[1,2-A]PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS BIOFOCUS DPI LTD (GB) 2013-01-30 EP disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
EP-2193131-A2 IMIDAZO[1,2-A]PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS Biofocus DPI Limited (GB) 2010-06-09 EP disclosed
WO-2009024585-A2 IMIDAZO [1,2-A] PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS BIOFOCUS DPI LIMITED (GB) 2009-02-26 WO disclosed
WO-2009024585-A2 IMIDAZO [1,2-A] PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS BIOFOCUS DPI LIMITED (GB) 2009-02-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS CYP3A5, HAVCR2, CYP3A43 SSTR4 2078/4885CCNE2 1676/4885CCNE1 1338/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.