SCHEMBL21812948

SCHEMBL21812948

O=C(O)NCc1nc(-c2cn[nH]c2)cs1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 6/20 0.42
ROCK2 O75116 8/20 0.41
KCNH2 Q12809 1/20 0.41
GRM4 Q14833 1/20 0.41
GPR35 Q9HC97 1/20 0.40
MAPK1 P28482 1/20 0.39
ROCK1 Q13464 2/20 0.37
ALDH1A1 P00352 1/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21812556 0.83 HDAC3 (0.48) NAMPTROCK2KCNH2GRM4ROCK1
SCHEMBL21834597 0.76 ALDH1A1 (0.49) ROCK2MAPK1ROCK1ALDH1A1RAB9A
SCHEMBL2342868 0.73 CNR2 (0.62) MAPK1ALDH1A1RAB9AL3MBTL1
SCHEMBL25180665 0.72 RAB9A (0.54) NAMPTMAPK1ALDH1A1RAB9A
SCHEMBL22501830 0.69 ROCK2 (0.59) ROCK2ROCK1
SCHEMBL19259693 0.68 ROCK2 (0.41) ROCK2MAPK1ALDH1A1RAB9A
SCHEMBL29999682 0.68 NPC1 (0.36) ALDH1A1RAB9AL3MBTL1
SCHEMBL29859845 0.68 KCNH2 (0.48) KCNH2GRM4MAPK1ALDH1A1RAB9A
SCHEMBL17293023 0.68 NAMPT (0.51) NAMPTROCK2
SCHEMBL18215350 0.68 MAPK1 (0.56) MAPK1ALDH1A1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020064175-A1 INDANE DERIVATIVES FOR USE IN THE TREATMENT OF BACTERIAL INFECTION ANTABIO SAS (FR) 2020-04-02 WO disclosed
EP-3628672-A1 INDANE DERIVATIVES FOR USE IN THE TREATMENT OF BACTERIAL INFECTION Antabio SAS (FR) 2020-04-01 EP disclosed