SCHEMBL21815216

SCHEMBL21815216

CCCC(=O)OC(=O)c1c[nH]nc1OCCCOCC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 8/20 0.37
CCNE1 P24864 8/20 0.37
CDK2 P24941 8/20 0.37
CCNB2 O95067 5/20 0.35
CDK1 P06493 5/20 0.35
CCNB1 P14635 5/20 0.35
CCNB3 Q8WWL7 5/20 0.35
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
CCND2 P30279 1/20 0.34
CCND3 P30281 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 2/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 4/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21815219 0.94 GRM4 (0.36) CCNE2CCNE1CDK2CCNB2CDK1
SCHEMBL21815215 0.89 CCNE2 (0.36) CCNE2CCNE1CDK2CCNB2CDK1
SCHEMBL21804283 0.83 TSHR (0.47) ALDH1A1TSHRL3MBTL1TDP1TP53
SCHEMBL21804494 0.76 TSHR (0.49) ALDH1A1HTTTSHR
SCHEMBL21815230 0.73 RARB (0.43) ALDH1A1HTTSMN1; SMN2TSHRMAPK1
SCHEMBL21805554 0.72 TSHR (0.47) ALDH1A1HTTTSHRL3MBTL1TDP1
SCHEMBL20523594 0.72 ALDH1A1 (0.33) CCNE2CCNE1CDK2ALDH1A1MAPK1
SCHEMBL7257515 0.70 ALDH1A1 (0.55) ALDH1A1TSHRL3MBTL1TDP1TP53
SCHEMBL28026639 0.68 LMNA (0.55) ALDH1A1SMN1; SMN2TSHRL3MBTL1TDP1
SCHEMBL11552370 0.68 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3856188-A1 AMINOPYRIMIDINE COMPOUND Cardurion Pharmaceuticals, LLC (US) 2021-08-04 EP disclosed
WO-2020068854-A1 AMINOPYRIMIDINE COMPOUND CARDURION PHARMACEUTICALS, LLC (US) 2020-04-02 WO disclosed