SCHEMBL21835593

SCHEMBL21835593

CON(C)C(=O)c1cc[nH]n1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38
CLK1 P49759 1/20 0.36
DYRK1A Q13627 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
TRPM8 Q7Z2W7 2/20 0.35
SLC6A3 Q01959 1/20 0.33
FAAH O00519 1/20 0.31
ICAM1 P05362 1/20 0.30
SELE P16581 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2078311 0.82 SMN1; SMN2 (0.39) MEN1KMT2ARAB9ADYRK1A
SCHEMBL20588923 0.79
SCHEMBL4307277 0.79
SCHEMBL3150437 0.77 KMT2A (0.34) MLYCDMEN1KMT2ARAB9AMAPK1
SCHEMBL28297724 0.76 CNR2 (0.44)
SCHEMBL5285523 0.76 ALDH1A1 (0.47) MLYCDMEN1KMT2ATDP1RAB9A
SCHEMBL10593163 0.75
Trimethylammonium SCHEMBL27464061 0.75 HCAR2 (0.39) TDP1MAPK1
SCHEMBL6003817 0.74 KDM4E (0.50) MEN1KMT2ARAB9A
SCHEMBL5167577 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12264138-B2 Process for the preparation of microbiocidal oxadiazole derivatives SYNGENTA CROP PROTECTION AG (CH) 2025-04-01 US disclosed
US-20240174683-A1 MAP4K1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2024-05-30 US disclosed
US-11945796-B2 Substituted pyridine derivatives as SARM1 inhibitors NURA BIO, INC. (US) 2024-04-02 US disclosed
EP-4288437-A1 MAP4K1 INHIBITORS Bayer Aktiengesellschaft (DE) 2023-12-13 EP disclosed
CN-116438171-A Substituted pyridine derivatives as SARM1 inhibitors 努拉生物公司 2023-07-14 CN disclosed
WO-2022167627-A1 MAP4K1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2022-08-11 WO disclosed
US-20220194907-A1 PROCESS FOR THE PREPARATION OF MICROBIOCIDAL OXADIAZOLE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2022-06-23 US disclosed
US-11358957-B2 Microbiocidal oxadiazole derivatives SYNGENTA PARTICIPATIONS AG (CH) 2022-06-14 US disclosed
US-20220081417-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS SARM1 INHIBITORS NURA BIO, INC. 2022-03-17 US disclosed
US-20220081417-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS SARM1 INHIBITORS NURA BIO, INC. 2022-03-17 US disclosed
US-20200277287-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2020-09-03 US disclosed
WO-2020068846-A1 HETEROCYCLIC COMPOUND HETEROCYCLIC COMPOUND (US) 2020-04-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11945796-B2 Substituted pyridine derivatives as SARM1 inhibitors SARM1, SARNP, ADRM1 MLYCD 2695/4885MEN1 4471/4885KMT2A 1817/4885
US-20220081417-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS SARM1 INHIBITORS SARM1, SARNP, ADRM1 MLYCD 2695/4885MEN1 4471/4885KMT2A 1817/4885
US-12264138-B2 Process for the preparation of microbiocidal oxadiazole derivatives CYP51A1, MPO, NOX5 MLYCD 466/4885MEN1 3852/4885KMT2A 4305/4885
US-20240174683-A1 MAP4K1 INHIBITORS MAP3K4, MAP4K4, MAP4K1 MLYCD 2451/4885MEN1 468/4885KMT2A 2250/4885
US-20200277287-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES PRF1, NOX1, ARG2 MLYCD 371/4885MEN1 3805/4885KMT2A 4506/4885
US-11358957-B2 Microbiocidal oxadiazole derivatives PRF1, NOX1, ARG2 MLYCD 371/4885MEN1 3805/4885KMT2A 4506/4885
US-20220194907-A1 PROCESS FOR THE PREPARATION OF MICROBIOCIDAL OXADIAZOLE DERIVATIVES CYP51A1, MPO, NOX5 MLYCD 466/4885MEN1 3852/4885KMT2A 4305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.