SCHEMBL2185490

SCHEMBL2185490

COc1ccc(-c2nc(C(=O)O)cc(N3CCCC3)n2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.49
ALDH1A1 P00352 6/20 0.49
HPGD P15428 5/20 0.49
GLA P06280 1/20 0.49
GAA P10253 1/20 0.49
HSD17B10 Q99714 2/20 0.49
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MAPT P10636 6/20 0.48
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
USP2 O75604 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2178164 0.89 MAPK1 (0.49) KDM4EALDH1A1HPGDGLAGAA
SCHEMBL12408682 0.81 L3MBTL1 (0.64) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL6394883 0.80 HPGD (0.63) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL2186195 0.80 KDM4E (0.70) KDM4EALDH1A1HPGDGLAGAA
SCHEMBL2927049 0.79 HPGD (0.67) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL2179510 0.79 MAPT (0.53) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL19072152 0.76 SCN9A (0.63) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL6395632 0.75 MAPT (0.57) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL19180309 0.74 ALDH1A1 (0.62) KDM4EALDH1A1HPGDGLAGAA
SCHEMBL2178587 0.71 KMT2A (0.59) KDM4EALDH1A1HPGDGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342191-A1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE Mitsubishi Tanabe Pharma Corporation (JP) 2011-07-13 EP disclosed
WO-2010030027-A1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2010-03-18 WO disclosed