SCHEMBL2185778

SCHEMBL2185778

CN(C(=O)c1ccsc1C(=O)O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.54
DHODH Q02127 1/20 0.47
KDM4E B2RXH2 2/20 0.46
KMT2A Q03164 1/20 0.46
MAOB P27338 1/20 0.44
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.41
ATM Q13315 1/20 0.41
LMNA P02545 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
EDNRA P25101 1/20 0.40
NR1H3 Q13133 1/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2186762 0.87 POLB (0.50) POLBDHODHKDM4EKMT2AMAOB
SCHEMBL2187905 0.84 L3MBTL1 (0.49) POLBKDM4EKMT2ALMNAALDH1A1
SCHEMBL2185780 0.80 POLB (0.50) POLBKDM4EKMT2AMAOBHTT
SCHEMBL2189405 0.78 KDM4E (0.49) POLBKDM4EKMT2AHTTLMNA
SCHEMBL9001638 0.78 POLB (0.75) POLBKDM4EKMT2AMAOBHTT
SCHEMBL69159 0.73 ALDH1A1 (0.58) POLBDHODHKDM4EKMT2ANPSR1
SCHEMBL5234734 0.73 HTT (0.41) POLBKDM4EKMT2AHTTALDH1A1
SCHEMBL2186765 0.73 KMT2A (0.43) POLBKDM4EKMT2AHTTNPSR1
SCHEMBL11129083 0.72 CES2 (0.53) POLBKDM4EKMT2AHTTLMNA
SCHEMBL3621051 0.72 DHODH (0.51) POLBDHODHKDM4EKMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578741-B1 AROMATIC COMPOUNDS AS ANTI-INFLAMMATORY, IMMUNOMODULATORY AND ANTI-PROLIFERATORY AGENTS 4SC AG (DE) 2011-07-13 EP claimed
EP-1578741-B1 AROMATIC COMPOUNDS AS ANTI-INFLAMMATORY, IMMUNOMODULATORY AND ANTI-PROLIFERATORY AGENTS 4SC AG (DE) 2011-07-13 EP disclosed