SCHEMBL21859488

SCHEMBL21859488

C#CC1C=CC(O[Si](C)(C)C(C)(C)C)[C@@H](CO)O1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 13/20 0.37
CYP2C19 P33261 12/20 0.37
CYP2C9 P11712 10/20 0.37
MAPT P10636 6/20 0.37
TP53 P04637 1/20 0.37
CYP2D6 P10635 3/20 0.36
ALDH1A1 P00352 6/20 0.34
TSHR P16473 3/20 0.34
HSD17B10 Q99714 1/20 0.33
MAPK1 P28482 1/20 0.32
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21832123 1.00 CYP3A4 (0.37) CYP3A4CYP2C19CYP2C9MAPTTP53
SCHEMBL21859489 0.84 ALDH1A1 (0.34) CYP2C19MAPTALDH1A1TSHR
SCHEMBL21832102 0.84 ALDH1A1 (0.34) CYP2C19MAPTALDH1A1TSHR
SCHEMBL21832122 0.74
SCHEMBL21859491 0.74
SCHEMBL21832116 0.71
SCHEMBL1578416 0.70 LGALS8 (0.37)
SCHEMBL16155602 0.70 LGALS8 (0.37)
SCHEMBL21859499 0.69
SCHEMBL24797484 0.68 CYP2C19 (0.53) CYP3A4CYP2C19MAPTCYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11191273-B2 Methods of making pyranopyrans such as pyranopyran nitrile and methods of using pyranopyrans such as pyranopyran nitrile THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF AGRICULTURE (US) 2021-12-07 US disclosed
US-20200093132-A1 Methods Of Making Pyranopyrans Such As Pyranopyran Nitrile And Methods of Using Pyranopyrans Such As Pyranopyran Nitrile VILLANOVA UNIVERSITY 2020-03-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200093132-A1 Methods Of Making Pyranopyrans Such As Pyranopyran Nitrile And Methods of Using Pyranopyrans Such As Pyranopyran Nitrile CBR1, NOX1, NOX3 CYP3A4 92/4885CYP2C19 325/4885CYP2C9 120/4885
US-11191273-B2 Methods of making pyranopyrans such as pyranopyran nitrile and methods of using pyranopyrans such as pyranopyran nitrile CBR1, NOX1, NOX3 CYP3A4 92/4885CYP2C19 325/4885CYP2C9 120/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.