SCHEMBL21859489

SCHEMBL21859489

C#CC1C=CC(O[Si](C)(C)C(C)(C)C)[C@@H](CO[Si](C)(C)C(C)(C)C)O1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.32
DUT P33316 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21832102 1.00 ALDH1A1 (0.34) ALDH1A1MAPTTSHRCYP2C19DUT
SCHEMBL21832123 0.84 CYP3A4 (0.37) ALDH1A1MAPTTSHRCYP2C19
SCHEMBL21859488 0.84 CYP3A4 (0.37) ALDH1A1MAPTTSHRCYP2C19
SCHEMBL24420699 0.76 DUT (0.33) DUT
SCHEMBL22639340 0.76 DUT (0.33) DUT
SCHEMBL22639184 0.76 DUT (0.33) DUT
SCHEMBL21859491 0.76
SCHEMBL21832122 0.76
SCHEMBL21698858 0.74 DUT (0.31) DUT
SCHEMBL21859500 0.70 TOP2A (0.31) DUT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11191273-B2 Methods of making pyranopyrans such as pyranopyran nitrile and methods of using pyranopyrans such as pyranopyran nitrile THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF AGRICULTURE (US) 2021-12-07 US disclosed
US-20200093132-A1 Methods Of Making Pyranopyrans Such As Pyranopyran Nitrile And Methods of Using Pyranopyrans Such As Pyranopyran Nitrile VILLANOVA UNIVERSITY 2020-03-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200093132-A1 Methods Of Making Pyranopyrans Such As Pyranopyran Nitrile And Methods of Using Pyranopyrans Such As Pyranopyran Nitrile CBR1, NOX1, NOX3 ALDH1A1 419/4885MAPT 4150/4885TSHR 1811/4885
US-11191273-B2 Methods of making pyranopyrans such as pyranopyran nitrile and methods of using pyranopyrans such as pyranopyran nitrile CBR1, NOX1, NOX3 ALDH1A1 419/4885MAPT 4150/4885TSHR 1811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.