SCHEMBL2186891

SCHEMBL2186891

COCCN1C(=O)c2c(O)c(=O)c(C(=O)NCc3ccc(F)c(OC)c3)cn2CC1O

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC22A2 O15244 10/20 0.44
CYP3A4 P08684 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2185191 0.90 SLC22A2 (0.46) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL2185146 0.89 P2RX7 (0.47) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL3523992 0.88 SLC22A2 (0.47) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL3528016 0.87 ALDH1A1 (0.43)
SCHEMBL2186951 0.86 SLC22A2 (0.41) SLC22A2
SCHEMBL2186319 0.85 SLC22A2 (0.53) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL3525535 0.84 PDE10A (0.42)
SCHEMBL3524286 0.84 ELANE (0.42) SLC22A2
SCHEMBL2186875 0.84 SLC22A2 (0.62) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL3525528 0.83 MAPK1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1852434-B1 BICYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITING ACTIVITY SHIONOGI & CO (JP) 2011-07-13 EP disclosed
US-7858788-B2 Bicyclic carbamoylpyridone derivative having HIV integrase inhibitory activity SHIONOGI & CO., LTD. (JP) 2010-12-28 US disclosed
EP-1852434-A1 BICYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITING ACTIVITY Shionogi Co., Ltd. (JP) 2007-11-07 EP disclosed