SCHEMBL2187677

SCHEMBL2187677

Cc1cc(CC(=O)NC(Cc2ccc(Oc3ccc(F)cc3)cc2)C(N)=O)[nH]n1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 15/20 0.48
GPR34 Q9UPC5 2/20 0.41
S1PR1 P21453 2/20 0.41
FPR2 P25090 2/20 0.39
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2185465 0.79 SCN9A (0.49) SCN9AFPR2CNR2
SCHEMBL2187665 0.78 S1PR1 (0.55) SCN9AS1PR1
SCHEMBL2171623 0.78 PTPN1 (0.57) SCN9AGPR34CNR2
SCHEMBL1371808 0.75 S1PR1 (0.73) SCN9AS1PR1
SCHEMBL2352923 0.75 SCN9A (0.64) SCN9AGPR34
SCHEMBL2357204 0.75 SCN9A (0.52) SCN9AGPR34
SCHEMBL2353034 0.74 SCN9A (0.48) SCN9AGPR34FPR2
SCHEMBL2172340 0.74 SCN9A (0.51) SCN9AGPR34FPR2
SCHEMBL2169958 0.73 SCN9A (0.47) SCN9ACNR2
SCHEMBL2171096 0.72 SCN9A (0.51) SCN9AGPR34

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed