SCHEMBL2169958

SCHEMBL2169958

CC(C)N1CCN(CC(=O)NC(Cc2ccc(Oc3ccc(F)cc3)cc2)C(N)=O)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.47
ALDH1A1 P00352 3/20 0.46
HRH3 Q9Y5N1 2/20 0.42
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
S1PR2 O95136 1/20 0.39
CNR2 P34972 1/20 0.39
STAT3 P40763 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171096 0.89 SCN9A (0.51) SCN9AALDH1A1MEN1KMT2A
SCHEMBL2170108 0.87 LMNA (0.52) SCN9AALDH1A1CA1CA2CA7
SCHEMBL2170146 0.86 SCN9A (0.48) SCN9AALDH1A1LMNAMEN1KMT2A
SCHEMBL2170398 0.86 ALDH1A1 (0.51) SCN9AALDH1A1CNR2
SCHEMBL2171621 0.86 QRFPR (0.50) SCN9AALDH1A1
SCHEMBL2171851 0.86 KMT2A (0.53) SCN9AALDH1A1KMT2A
SCHEMBL2169808 0.86 SCN9A (0.48) SCN9AALDH1A1
SCHEMBL2356486 0.85 SCN9A (0.45) SCN9AALDH1A1S1PR2
SCHEMBL2171705 0.85 MEN1 (0.60) ALDH1A1CA1CA2CA7CA9
SCHEMBL2170811 0.84 MAPT (0.54) SCN9AALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed