SCHEMBL21882076

SCHEMBL21882076

CC(C)(C)OC(=O)NC1CCN(N=O)CC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.55
BTK Q06187 1/20 0.48
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
HSD11B1 P28845 3/20 0.46
CYP2C9 P11712 1/20 0.46
EPHX1 P07099 2/20 0.46
KCNA3 P22001 1/20 0.44
CKS1B P61024 1/20 0.44
SKP1 P63208 1/20 0.44
SKP2 Q13309 1/20 0.44
GAA P10253 2/20 0.43
DRD2 P14416 2/20 0.43
NAMPT P43490 1/20 0.42
KDM1A O60341 1/20 0.42
MAOB P27338 1/20 0.42
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23119939 0.91 CTSK (0.59) CTSKBTKCA1CA2HSD11B1
SCHEMBL28830472 0.91 CTSK (0.59) CTSKBTKCA1CA2HSD11B1
SCHEMBL28830439 0.91 CTSK (0.59) CTSKBTKCA1CA2HSD11B1
SCHEMBL28830425 0.83 CTSK (0.50) CTSKBTKCA1CA2HSD11B1
SCHEMBL31317827 0.82 CA1 (0.59) CTSKBTKCA1CA2HSD11B1
SCHEMBL17951138 0.82 CA1 (0.59) CTSKBTKCA1CA2HSD11B1
SCHEMBL31317808 0.82 CA1 (0.59) CTSKBTKCA1CA2HSD11B1
SCHEMBL359203 0.81 CTSK (0.59) CTSKBTKCA1CA2HSD11B1
SCHEMBL24068416 0.81 CTSK (0.59) CTSKBTKCA1CA2HSD11B1
SCHEMBL3702152 0.80 BTK (0.61) CTSKBTKCA1CA2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025011633-A1 ANTAGONIST OF MAS-RELATED G PROTEIN-COUPLED RECEPTOR X2 AND USE THEREOF 北京普祺医药科技股份有限公司 2025-01-16 WO disclosed
US-20220071966-A1 INHIBITORS OF INTEGRATED STRESS RESPONSE PATHWAY Praxis Biotech LLC 2022-03-10 US disclosed
US-11166942-B2 Inhibitors of integrated stress response pathway Praxis Biotech LLC (US) 2021-11-09 US disclosed
US-20200101047-A1 INHIBITORS OF INTEGRATED STRESS RESPONSE PATHWAY Praxis Biotech LLC 2020-04-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11166942-B2 Inhibitors of integrated stress response pathway ATF4, DDIT3, ATF1 CTSK 3839/4885BTK 1436/4885CA1 4637/4885
US-20220071966-A1 INHIBITORS OF INTEGRATED STRESS RESPONSE PATHWAY ATF4, DDIT3, ATF1 CTSK 3839/4885BTK 1436/4885CA1 4637/4885
US-20200101047-A1 INHIBITORS OF INTEGRATED STRESS RESPONSE PATHWAY ATF4, DDIT3, ATF1 CTSK 3839/4885BTK 1436/4885CA1 4637/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.