SCHEMBL21883433

SCHEMBL21883433

CC(C)CC(NC(=O)CNC(=O)C(N)Cc1ccccc1)C(=O)NC(CCCN)C(N)=O

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 9/20 0.57
OPRM1 P35372 5/20 0.57
OPRK1 P41145 5/20 0.57
KISS1R Q969F8 1/20 0.56
CTSB P07858 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27898271 0.90 OPRD1 (0.61) OPRD1OPRM1OPRK1
SCHEMBL31736791 0.89 OPRK1 (0.57) OPRD1OPRM1OPRK1
SCHEMBL24152321 0.86 MMP2 (0.54) OPRD1OPRM1OPRK1
SCHEMBL29871918 0.86 NPY4R (0.66) OPRD1OPRM1OPRK1KISS1R
SCHEMBL31433318 0.85 OPRD1 (0.58) OPRD1OPRM1OPRK1CTSB
SCHEMBL18176630 0.84 KISS1R (0.62) OPRD1OPRM1OPRK1KISS1R
SCHEMBL21886335 0.84 KISS1R (0.62) OPRD1OPRM1OPRK1KISS1R
SCHEMBL11931977 0.84 KISS1R (0.62) OPRD1OPRM1OPRK1KISS1R
SCHEMBL19249634 0.84 KISS1R (0.62) OPRD1OPRM1OPRK1KISS1R
SCHEMBL29568724 0.84 OPRK1 (0.59) OPRD1OPRM1OPRK1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020056249-A1 ORAL FORMULATIONS OF KAPPA OPIOID RECEPTOR AGONISTS CARA THERAPEUTICS, INC. (US) 2020-03-19 WO disclosed