SCHEMBL21887872

SCHEMBL21887872

CC1Cn2nc(C(=O)NCC(F)(F)F)cc2-c2ccc(-c3cccc(S(C)(=O)=O)c3)cc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.39
IDH2 P48735 1/20 0.38
PIK3CD O00329 1/20 0.36
PIK3CG P48736 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
KLKB1 P03952 2/20 0.36
RXRA P19793 3/20 0.35
NR1H3 Q13133 3/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
DPP4 P27487 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21887770 0.85 NR1H2 (0.39) NR1H2RXRANR1H3JAK2JAK1
SCHEMBL21887871 0.84 NR1H2 (0.43) NR1H2PIK3CDPIK3CGRXRANR1H3
SCHEMBL21888599 0.79 NR1H2 (0.44) NR1H2PIK3CDPIK3CGRXRANR1H3
SCHEMBL21887739 0.76 NR1H2 (0.53) NR1H2PIK3CDPIK3CGRXRANR1H3
SCHEMBL3472767 0.76 NR1H2 (0.45) NR1H2IDH2CTSLCTSBCTSS
SCHEMBL16553538 0.75 NR1H2 (0.67) NR1H2IDH2PIK3CDPIK3CGCTSL
SCHEMBL3472382 0.71 NR1H2 (0.46) NR1H2IDH2CTSLCTSBCTSS
SCHEMBL16126467 0.69 NR1H2 (0.41) NR1H2IDH2RXRANR1H3CHRNB2
SCHEMBL3473255 0.68 NR1H2 (0.69) NR1H2IDH2RXRANR1H3
SCHEMBL3470791 0.68 RXRA (0.73) NR1H2IDH2RXRANR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3626712-A2 LIVER X RECEPTOR (LXR) MODULATORS Ellora Therapeutics, Inc. (US) 2020-03-25 EP disclosed