SCHEMBL2190249

SCHEMBL2190249

Fc1cc(Nc2ccc(Oc3ccccc3)cc2)ccn1.OCCNc1cc(Nc2ccc(Oc3ccccc3)cc2)ccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.42
ADRA1D P25100 2/20 0.42
HTR2C P28335 2/20 0.42
ADRA1A P35348 2/20 0.42
ADRA1B P35368 2/20 0.42
DRD2 P14416 1/20 0.42
P2RX3 P56373 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
JAK3 P52333 1/20 0.41
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
ERBB2 P04626 1/20 0.39
SCN9A Q15858 1/20 0.39
KCNH3 Q9ULD8 1/20 0.39
ACVRL1 P37023 1/20 0.39
BRAF P15056 1/20 0.38
KDR P35968 1/20 0.38
MAPK14 Q16539 1/20 0.38
TNNI3K Q59H18 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2174904 0.93 HTR7 (0.46) HTR7ADRA1DHTR2CADRA1AADRA1B
SCHEMBL2174129 0.84 SCN9A (0.51) JAK2JAK1JAK3ERBB2SCN9A
SCHEMBL2177165 0.78 ALDH1A1 (0.52) P2RX3GAAKMT2A
SCHEMBL2177484 0.77 EGFR (0.57) GAAKMT2ASCN9ABRAFKDR
SCHEMBL8287302 0.75 AURKA (0.51) KMT2ASCN9AKCNH3
SCHEMBL13977412 0.75 EGFR (0.44) JAK2GAAACVRL1KDR
SCHEMBL2176931 0.72 SCN9A (0.50) GAAKMT2ASCN9AKCNH3
SCHEMBL2174899 0.72 PLK1 (0.46) HTR7ADRA1DHTR2CADRA1AADRA1B
SCHEMBL2173982 0.68 RAB9A (0.57) GAAKMT2AKCNH3
SCHEMBL31580872 0.68 BRAF (0.48) P2RX3KMT2AERBB2SCN9AACVRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2519501-A2 SUBSTITUTED PYRIDINES AND PYRIMIDINES FOR THE PRODUCTION OF CARDIOMYOCYTE-LIKE CELLS Technische Universität Wien (AT) 2012-11-07 EP disclosed
WO-2011079343-A2 SUBSTITUTED PYRIDINES AND PYRIMIDINES TECHNISCHE UNIVERSITAET WIEN (AT) 2011-07-07 WO disclosed