SCHEMBL2174899

SCHEMBL2174899

CC(O)Nc1cc(Nc2ccc(Oc3ccccc3)cc2)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.46
HTR7 P34969 3/20 0.46
GCK P35557 1/20 0.45
SCN9A Q15858 2/20 0.44
ERBB2 P04626 1/20 0.44
ACVRL1 P37023 1/20 0.43
MAPKAPK2 P49137 2/20 0.43
ADRA1D P25100 1/20 0.42
HTR2C P28335 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
FGFR2 P21802 2/20 0.42
KCNH2 Q12809 1/20 0.40
SCN5A Q14524 1/20 0.40
HTT P42858 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2174904 0.77 HTR7 (0.46) HTR7GCKSCN9AERBB2ACVRL1
SCHEMBL2174129 0.74 SCN9A (0.51) SCN9AERBB2FGFR2KCNH2SCN5A
SCHEMBL31580872 0.73 BRAF (0.48) GCKSCN9AERBB2ACVRL1HTT
SCHEMBL2190249 0.72 HTR7 (0.42) HTR7GCKSCN9AERBB2ACVRL1
SCHEMBL30046984 0.70 KDR (0.54) SCN9AERBB2SCN5AHTTALDH1A1
SCHEMBL14435643 0.70 LTA4H (0.63) SCN9AERBB2SCN5AHTTALDH1A1
SCHEMBL17948198 0.70 LTA4H (0.63) SCN9AERBB2SCN5AHTTALDH1A1
SCHEMBL24178149 0.70
SCHEMBL18657532 0.69 ALDH1A1 (0.67) SCN9AERBB2SCN5AALDH1A1HPGD
SCHEMBL29066282 0.69 ACVRL1 (0.61) ACVRL1MAPKAPK2ALDH1A1ALOX12KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079343-A2 SUBSTITUTED PYRIDINES AND PYRIMIDINES TECHNISCHE UNIVERSITAET WIEN (AT) 2011-07-07 WO disclosed