SCHEMBL21936743

SCHEMBL21936743

Cc1ccc2c(c1)CN(C)N=C2

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 10/20 0.35
SLC6A4 P31645 10/20 0.35
SLC6A3 Q01959 10/20 0.35
CYP2D6 P10635 1/20 0.32
HSD17B10 Q99714 1/20 0.31
SRD5A1 P18405 1/20 0.30
HTR5A P47898 1/20 0.30
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27103162 0.85 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3HSD17B10HTR5A
SCHEMBL29710439 0.75 TRPA1 (0.38) SLC6A2SLC6A4SLC6A3CYP2D6NOTUM
SCHEMBL11441366 0.75 TRPA1 (0.38) SLC6A2SLC6A4SLC6A3CYP2D6NOTUM
SCHEMBL28162719 0.69 KDM4E (0.33)
SCHEMBL255505 0.68 HTR5A (0.37) HTR5ANOTUM
SCHEMBL8340988 0.68 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3CYP2D6HSD17B10
SCHEMBL30025550 0.65 ADRA2A (0.34) HTR5ANOTUM
SCHEMBL7938077 0.65 ADRA2A (0.34) HTR5ANOTUM
Hydrochloric Acid SCHEMBL11820690 0.64 ADRA2A (0.33) HTR5ANOTUM
SCHEMBL2835665 0.63 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3633380-A1 METHOD FOR PREDICTING THERAPEUTIC EFFECT OF LSD1 INHIBITOR BASED ON EXPRESSION OF INSM1 Taiho Pharmaceutical Co., Ltd. (JP) 2020-04-08 EP disclosed