SCHEMBL21940485

SCHEMBL21940485

COc1cc(C#N)nnc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
PDE5A O76074 7/20 0.38
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NQO1 P15559 1/20 0.35
MAPT P10636 2/20 0.35
KMT2A Q03164 1/20 0.35
PDE10A Q9Y233 1/20 0.35
CHEK1 O14757 3/20 0.35
ALDH1A1 P00352 2/20 0.34
USP2 O75604 1/20 0.34
PGK1 P00558 1/20 0.33
HPGD P15428 1/20 0.33
IKBKB O14920 1/20 0.33
AURKA O14965 1/20 0.33
DCLK1 O15075 1/20 0.33
RPS6KA5 O75582 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
RET P07949 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20606943 0.74 ALDH1A1 (0.37) KDM4EL3MBTL1MAPTKMT2AALDH1A1
SCHEMBL2047755 0.73 ALDH1A1 (0.45) KDM4EL3MBTL1KMT2AALDH1A1PGK1
SCHEMBL29549875 0.73 ALDH1A1 (0.45) KDM4EL3MBTL1KMT2AALDH1A1PGK1
SCHEMBL14135244 0.73 KMO (0.34)
SCHEMBL29549876 0.73 ALDH1A1 (0.45) KDM4EL3MBTL1KMT2AALDH1A1PGK1
SCHEMBL12093320 0.71 PGK1 (0.36) KDM4EL3MBTL1MAPTALDH1A1PGK1
SCHEMBL22042633 0.69 CYP3A4 (0.37) KDM4EL3MBTL1MAPTALDH1A1PGK1
SCHEMBL15687643 0.69 GAA (0.42) KDM4EPDE5AL3MBTL1ALDH1A1PGK1
SCHEMBL21940288 0.69 ALDH1A1 (0.35) KDM4EMAPTKMT2AALDH1A1HPGD
SCHEMBL10368496 0.69 NOTUM (0.31) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423445-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2020-04-01 EP disclosed