SCHEMBL21961391

SCHEMBL21961391

ONc1cn[nH]c1C1CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 3/20 0.44
MAPK8 P45983 3/20 0.35
MAPK9 P45984 3/20 0.35
MAPK10 P53779 3/20 0.35
CDK2 P24941 3/20 0.35
GSK3B P49841 2/20 0.35
MAP2K7 O14733 1/20 0.35
IKBKB O14920 1/20 0.35
MAPK13 O15264 1/20 0.35
MAP2K4 P45985 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
MAP2K6 P52564 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK14 Q16539 1/20 0.35
HCAR2 Q8TDS4 1/20 0.33
ACVR1 Q04771 1/20 0.32
TRPV1 Q8NER1 4/20 0.31
CCNA2 P20248 2/20 0.30
CDK1 P06493 1/20 0.30
CDK4 P11802 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21961392 0.77 HPGDS (0.38) HPGDSMAPK8MAPK9MAPK10CDK2
SCHEMBL14387558 0.68
SCHEMBL16531513 0.68
SCHEMBL21816205 0.67 HCAR2 (0.43) HPGDSMAPK8MAPK9MAPK10HCAR2
SCHEMBL23344298 0.64 GAA (0.41) HPGDSACVR1
SCHEMBL21849265 0.64 HPGDS (0.40) HPGDSMAPK8MAPK9MAPK10CDK2
SCHEMBL21964550 0.61 LMNA (0.33) CDK2CCNA2CDK1CDK4CCNB1
SCHEMBL22553834 0.56 MAPK8 (0.41) HPGDSMAPK8MAPK9MAPK10CDK2
SCHEMBL2568371 0.55
SCHEMBL16964472 0.55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3478675-B1 HETEROAROMATIC DERIVATIVES AS NIK INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2020-04-22 EP disclosed