SCHEMBL21962491

SCHEMBL21962491

COC[C@@H]1CCCN1c1ncc(C(=O)c2cccc(S(=O)(=O)C(F)(F)F)c2)s1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.39
ADORA2A P29274 6/20 0.39
ADORA1 P30542 6/20 0.39
FFAR2 O15552 1/20 0.36
FPR1 P21462 1/20 0.36
FPR2 P25090 1/20 0.36
CRHR1 P34998 1/20 0.36
TIPARP Q7Z3E1 1/20 0.36
ADRA1A P35348 3/20 0.35
MAP4K1 Q92918 1/20 0.35
SYK P43405 1/20 0.35
SCN9A Q15858 1/20 0.35
MAP3K12 Q12852 1/20 0.35
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22020076 1.00 VNN1 (0.39) VNN1ADORA2AADORA1FFAR2FPR1
SCHEMBL22019323 0.90 VNN1 (0.39) VNN1ADORA2AADORA1
SCHEMBL21962563 0.90 VNN1 (0.39) VNN1ADORA2AADORA1
SCHEMBL22020081 0.84 HSD11B1 (0.38) VNN1
SCHEMBL21962810 0.80 VNN1 (0.39) VNN1
SCHEMBL22020078 0.80 VNN1 (0.39) VNN1
SCHEMBL21962580 0.79 HDAC3 (0.43)
SCHEMBL22019142 0.77 VNN1 (0.38) VNN1
SCHEMBL21962621 0.77 VNN1 (0.38) VNN1
SCHEMBL21962619 0.77 SCD (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO claimed
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed