SCHEMBL21962552

SCHEMBL21962552

O=C(c1cccc(C(F)(F)F)c1)c1cnc(N2CCC[C@H](O)C2)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 4/20 0.48
VNN1 O95497 1/20 0.47
LMNA P02545 4/20 0.44
SCD O00767 1/20 0.43
KDM4E B2RXH2 2/20 0.42
USP2 O75604 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HPGD P15428 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
RAF1 P04049 1/20 0.41
BRAF P15056 1/20 0.41
MLYCD O95822 1/20 0.41
HDAC3 O15379 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962446 0.94 SCD (0.46) IDH2VNN1SCDKDM4EHPGD
SCHEMBL22019585 0.90 VNN1 (0.44) VNN1LMNASCDKDM4EUSP2
SCHEMBL21962851 0.90 VNN1 (0.44) VNN1LMNASCDKDM4EUSP2
SCHEMBL22019152 0.89 VNN1 (0.44) VNN1LMNASCDKDM4EUSP2
SCHEMBL21962681 0.89 VNN1 (0.44) VNN1LMNASCDKDM4EUSP2
SCHEMBL21962674 0.88 SCD (0.47) IDH2VNN1LMNASCDKDM4E
SCHEMBL21962568 0.87 LMNA (0.51) LMNASCDKDM4EHSD17B10HPGD
SCHEMBL21962779 0.87 MLYCD (0.49) LMNASCDKDM4EHSD17B10HPGD
SCHEMBL22019150 0.87 SCD (0.47) VNN1LMNASCDKDM4EUSP2
SCHEMBL22019591 0.86 LMNA (0.53) LMNASCDKDM4EHPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO claimed
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed