SCHEMBL21993358

SCHEMBL21993358

Bc1nc2cc(N(C)C(=O)C(Cc3cc(F)cc(F)c3)N(C)C(=O)OC(C)(C)C)ccc2s1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.39
AAK1 Q2M2I8 3/20 0.33
ADORA1 P30542 1/20 0.33
CLK1 P49759 1/20 0.32
CLK2 P49760 1/20 0.32
DYRK1A Q13627 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21992663 0.81 ADORA1 (0.33) PAX8AAK1ADORA1
SCHEMBL21992599 0.80 DYRK1A (0.35) AAK1CLK1CLK2DYRK1A
SCHEMBL19969184 0.80 DYRK1A (0.35) AAK1CLK1CLK2DYRK1A
SCHEMBL19969330 0.80 PAX8 (0.55) PAX8DYRK1A
SCHEMBL21992592 0.79 KMT2A (0.35) PAX8AAK1ADORA1
SCHEMBL18180190 0.78 AAK1 (0.34) PAX8AAK1ADORA1
SCHEMBL21993352 0.78 AAK1 (0.34) PAX8AAK1ADORA1
SCHEMBL21992548 0.76 HDAC1 (0.35) PAX8AAK1ADORA1
SCHEMBL18180346 0.76 USP30 (0.33) PAX8AAK1ADORA1
SCHEMBL21993350 0.76 STAT3 (0.35) PAX8AAK1ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286166-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2020-05-13 EP disclosed