SCHEMBL21994450

SCHEMBL21994450

COc1ccc(Cc2[nH]nc(C(F)(F)F)c2C(N)=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.42
GFER P55789 1/20 0.42
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SAE1 Q9UBE0 1/20 0.38
UBA2 Q9UBT2 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PARP1 P09874 1/20 0.38
PARP10 Q53GL7 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
PARP4 Q9UKK3 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MPI P34949 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
GRM2 Q14416 1/20 0.38
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
VNN1 O95497 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21994369 0.79 ALDH1A1 (0.40) ALDH1A1MEN1KMT2AKDM4EMPI
SCHEMBL8662301 0.70 PARP10 (0.42) GAAALDH1A1MEN1KMT2ASAE1
SCHEMBL28173058 0.70 ALDH1A1 (0.44) GAAALDH1A1MEN1KMT2AKDM4E
SCHEMBL1754055 0.70 ALDH1A1 (0.42) ALDH1A1MEN1KMT2AKDM4EMPI
SCHEMBL8887688 0.68 ADORA3 (0.45) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL27370090 0.68 AURKA (0.39) GAAALDH1A1MEN1KMT2AKDM4E
SCHEMBL8213818 0.66 PARP10 (0.78) ALDH1A1KMT2ASAE1UBA2CA1
SCHEMBL20521837 0.66 GAA (0.53) GAAGRM2
SCHEMBL3468087 0.65 SLC5A2 (0.56) ALDH1A1KDM4EMPIAPOBEC3G
SCHEMBL30365897 0.65 ALDH1A1 (0.54) ALDH1A1MEN1KMT2ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3887371-A1 ARYL COMPOUNDS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTION F. Hoffmann-La Roche AG (CH) 2021-10-06 EP disclosed
WO-2020109191-A1 ARYL COMPOUNDS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTION F. HOFFMANN-LA ROCHE AG (CH) 2020-06-04 WO disclosed