SCHEMBL21995195

SCHEMBL21995195

O=C(O)NC(C(=O)NCc1ccc(CNC(=O)C(NC(=O)O)c2ccccc2)cc1)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
F2 P00734 2/20 0.56
F10 P00742 2/20 0.56
PRSS1 P07477 2/20 0.56
PKM P14618 1/20 0.55
POLB P06746 1/20 0.51
MTTP P55157 1/20 0.50
GPR88 Q9GZN0 1/20 0.49
GAA P10253 1/20 0.48
ERCC1 P07992 1/20 0.48
ERCC4 Q92889 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4793272 0.97 KMT2A (0.56) MEN1KMT2AF2F10PRSS1
SCHEMBL12168558 0.85 MEN1 (0.68) MEN1KMT2AF2F10PRSS1
SCHEMBL12168556 0.84 CA12 (0.61) MEN1KMT2AF2F10PRSS1
SCHEMBL24304020 0.81 KMT2A (0.54) MEN1KMT2AF2F10PRSS1
SCHEMBL30475545 0.80 CTSL (0.48) MEN1KMT2AF2F10PRSS1
SCHEMBL23715929 0.80 KMT2A (0.56) MEN1KMT2APKMGPR88GAA
SCHEMBL29527526 0.80 CTSS (0.73) MEN1KMT2AF2F10PRSS1
SCHEMBL6225123 0.79 F2 (0.50) MEN1KMT2AF2F10PRSS1
SCHEMBL6184348 0.79 CTSS (0.68)
SCHEMBL19471121 0.79 CTSS (0.50) MEN1KMT2AF2F10PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4342473-A2 COMPOUNDS USEFUL IN HIV THERAPY GlaxoSmithKline Intellectual Property Development Limited (GB) 2024-03-27 EP disclosed
US-20240051972-A1 Compounds Useful in HIV Therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2024-02-15 US disclosed
US-11873310-B2 Compounds useful in HIV therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2024-01-16 US disclosed
US-11492361-B2 Compounds useful in HIV therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-11-08 US disclosed
US-20220119417-A1 Compounds Useful in HIV Therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-04-21 US disclosed
EP-3886987-A1 COMPOUNDS USEFUL IN HIV THERAPY GlaxoSmithKline Intellectual Property Development Ltd (GB) 2021-10-06 EP disclosed
US-20210009609-A1 Compounds Useful in HIV Therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2021-01-14 US disclosed
US-10870663-B2 Compounds useful in HIV therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-12-22 US disclosed
US-20200299309-A1 Compounds Useful in HIV Therapy GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-09-24 US disclosed
WO-2020110056-A1 COMPOUNDS USEFUL IN HIV THERAPY GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-06-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220119417-A1 Compounds Useful in HIV Therapy CD4, CCR5, ABCB1 MEN1 3875/4885KMT2A 4288/4885F2 1434/4885
US-20240051972-A1 Compounds Useful in HIV Therapy CD4, CCR5, ABCB1 MEN1 3875/4885KMT2A 4288/4885F2 1434/4885
US-11873310-B2 Compounds useful in HIV therapy CD4, CCR5, ABCB1 MEN1 3875/4885KMT2A 4288/4885F2 1434/4885
US-10870663-B2 Compounds useful in HIV therapy CCR5, SLC11A2, CD4 MEN1 3938/4885KMT2A 2588/4885F2 2403/4885
US-11492361-B2 Compounds useful in HIV therapy CD4, CCR5, ABCB1 MEN1 3640/4885KMT2A 3866/4885F2 1482/4885
US-20200299309-A1 Compounds Useful in HIV Therapy CCR5, SLC11A2, CD4 MEN1 3938/4885KMT2A 2588/4885F2 2403/4885
US-20210009609-A1 Compounds Useful in HIV Therapy CD4, CCR5, ABCB1 MEN1 3640/4885KMT2A 3866/4885F2 1482/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.