SCHEMBL21996211

SCHEMBL21996211

COc1ccc(COC(C)CC=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.46
AGXT P21549 2/20 0.46
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SLC6A4 P31645 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42
APP P05067 3/20 0.41
HTT P42858 2/20 0.41
LDHA P00338 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 2/20 0.41
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
ALOX12 P18054 1/20 0.41
POLB P06746 1/20 0.41
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12772124 1.00 IDO1 (0.46) IDO1AGXTNPC1RAB9ASLC6A4
SCHEMBL13149244 0.83 ALDH1A1 (0.53) IDO1AGXTSLC6A4APPSMN1; SMN2
SCHEMBL31388986 0.83 ALDH1A1 (0.53) IDO1AGXTSLC6A4APPSMN1; SMN2
SCHEMBL12772128 0.81 CA1 (0.40) IDO1AGXTNPC1RAB9ASLC6A4
SCHEMBL11577777 0.81 SLC1A3 (0.45) IDO1TAAR1HTTALDH1A1TSHR
SCHEMBL13149138 0.81 IDO1 (0.47) IDO1AGXTSLC6A4APPSMN1; SMN2
SCHEMBL12770001 0.80 IDO1 (0.42) IDO1AGXTNPC1RAB9ASLC6A4
SCHEMBL7069810 0.79 IDO1 (0.48) IDO1AGXTNPC1RAB9ASLC6A4
SCHEMBL16594094 0.79 IDO1 (0.48) IDO1AGXTNPC1RAB9ASLC6A4
SCHEMBL28885907 0.79 IDO1 (0.52) IDO1AGXTSLC6A4APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12037354-B2 Cyclic pantetheine derivatives and uses thereof VECTIVBIO COMET AG (CH) 2024-07-16 US disclosed
US-20230107216-A1 PANTETHEINE DERIVATIVES AND USES THEREOF VECTIVBIO COMET AG, F/K/A COMET THERAPEUTICS, INC. (CH) 2023-04-06 US disclosed
US-20230072313-A1 CYCLIC PANTETHEINE DERIVATIVES AND USES THEREOF VECTIVBIO COMET AG, F/K/A COMET THERAPEUTICS, INC. (CH) 2023-03-09 US disclosed
CN-114478528-A Aroyl-substituted tricyclic compound, preparation method and application thereof 劲方医药科技(上海)有限公司 2022-05-13 CN disclosed
CN-113727966-A Panthenol derivatives and use thereof 彗星医疗股份有限公司 2021-11-30 CN disclosed
CN-113727986-A Cyclic panthenol derivative and use thereof 彗星医疗股份有限公司 2021-11-30 CN disclosed
EP-3887353-A1 PANTETHEINE DERIVATIVES AND USES THEREOF Comet Therapeutics, Inc. (US) 2021-10-06 EP disclosed
EP-3887381-A2 CYCLIC PANTETHEINE DERIVATIVES AND USES THEREOF Comet Therapeutics, Inc. (US) 2021-10-06 EP disclosed
WO-2020113209-A1 PANTETHEINE DERIVATIVES AND USES THEREOF COMET THERAPEUTICS, INC. (US) 2020-06-04 WO disclosed
WO-2020113213-A2 CYCLIC PANTETHEINE DERIVATIVES AND USES THEREOF COMET THERAPEUTICS, INC. (US) 2020-06-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230107216-A1 PANTETHEINE DERIVATIVES AND USES THEREOF VNN1, NQO1, VKORC1 IDO1 3671/4885AGXT 1353/4885NPC1 329/4885
US-20230072313-A1 CYCLIC PANTETHEINE DERIVATIVES AND USES THEREOF VNN1, VKORC1, PANK3 IDO1 3810/4885AGXT 2078/4885NPC1 581/4885
US-12037354-B2 Cyclic pantetheine derivatives and uses thereof VNN1, VKORC1, PANK3 IDO1 3810/4885AGXT 2078/4885NPC1 581/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.