SCHEMBL2199716

SCHEMBL2199716

C[C@@H](c1ccc(C(O)C(C)(C)N(C)C)cc1)N(C(=O)O)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.41
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
MTOR P42345 1/20 0.32
ALOX5 P09917 3/20 0.32
KDM4E B2RXH2 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2196089 0.84 AOC3 (0.42) AOC3ALDH1A1ALOX5KDM4EMEN1
SCHEMBL2197829 0.81 MTOR (0.31) AOC3MTORALOX5
SCHEMBL2429212 0.79 ESR1 (0.42) ALDH1A1HSD17B10ALOX5
SCHEMBL1448846 0.79 ESR1 (0.42) ALDH1A1HSD17B10ALOX5
SCHEMBL2197629 0.78 KDM4E (0.43) AOC3ALDH1A1HSD17B10KDM4EMEN1
SCHEMBL1270470 0.78 ALOX5 (0.51) ALDH1A1ALOX5MEN1KMT2ASMN1; SMN2
SCHEMBL2197076 0.78 ALOX5 (0.51) ALDH1A1ALOX5MEN1KMT2ASMN1; SMN2
SCHEMBL2576026 0.78 ALOX5 (0.51) ALDH1A1ALOX5MEN1KMT2ASMN1; SMN2
SCHEMBL2195384 0.77 RIPK1 (0.37) AOC3TSHRALOX5KDM4EMEN1
SCHEMBL2197771 0.77 PTGS2 (0.38) ALDH1A1TSHRALOX5KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977336-B2 Aminopyrimidine derivatives as PLK1 inhibitors BANYU PHARMACEUTICAL CO. LTD (JP) 2011-07-12 US disclosed