SCHEMBL22010661

SCHEMBL22010661

CCOC(=O)CNC(=O)C1(C)CCN(C)CC1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.41
EPHX2 P34913 1/20 0.40
OPRM1 P35372 6/20 0.40
PPID Q08752 3/20 0.40
SLC22A1 O15245 1/20 0.40
SLC6A4 P31645 1/20 0.40
ADRA1A P35348 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
KCNH2 Q12809 1/20 0.40
PPIB P23284 1/20 0.40
PPIA P62937 1/20 0.40
PPIG Q13427 1/20 0.40
NLRP3 Q96P20 2/20 0.37
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11038014 0.83 GAA (0.45) GAAEPHX2PPIDPPIBPPIA
SCHEMBL22172283 0.79 KMT2A (0.41) OPRM1SLC22A1SLC6A4ADRA1AOPRD1
SCHEMBL580416 0.75 EPHX2 (0.43) GAAEPHX2PPIDPPIBPPIA
SCHEMBL2607180 0.75 OPRM1 (0.54) OPRM1SLC22A1SLC6A4ADRA1AOPRD1
Iodide SCHEMBL30309825 0.74 OPRM1 (0.53) OPRM1SLC22A1SLC6A4ADRA1AOPRD1
SCHEMBL10053026 0.73 GAA (0.49) GAAMGAMSIMGAM2
SCHEMBL20069764 0.73 JAK2 (0.42)
SCHEMBL15232250 0.72 OPRM1 (0.44) GAAOPRM1SLC22A1SLC6A4ADRA1A
SCHEMBL20069677 0.71 CYP2C19 (0.46)
SCHEMBL18390115 0.71 RET (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020099882-A1 HETEROCYCLIC SPIRO-COMPOUNDS AS AM2 RECEPTOR INHIBITORS THE UNIVERSITY OF SHEFFIELD (GB) 2020-05-22 WO disclosed