SCHEMBL22012874

SCHEMBL22012874

C[C@@H]1Cc2cc(Br)ccc2C1=O

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 2/20 0.56
ACHE P22303 12/20 0.56
PBRM1 Q86U86 1/20 0.42
TDP2 O95551 1/20 0.42
PARP10 Q53GL7 1/20 0.42
PARP11 Q9NR21 1/20 0.42
ADRA2A P08913 1/20 0.42
PNMT P11086 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
S100A4 P26447 1/20 0.41
BCL2 P10415 1/20 0.39
MCL1 Q07820 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1500072 1.00 METAP1 (0.56) METAP1ACHEPBRM1TDP2PARP10
SCHEMBL29980313 0.85 ACHE (0.66) METAP1ACHEPBRM1PARP10ADRA2A
SCHEMBL6475805 0.85 ACHE (0.66) METAP1ACHEPBRM1PARP10ADRA2A
SCHEMBL10687118 0.82 PARP10 (0.47) METAP1ACHEPBRM1TDP2PARP10
SCHEMBL10687696 0.80 PARP10 (0.45) METAP1ACHEPBRM1TDP2PARP10
SCHEMBL2484416 0.79 ACHE (0.73) METAP1ACHEPARP10PARP11
SCHEMBL8555030 0.79 METAP1 (0.54) METAP1PBRM1TDP2PARP10PARP11
SCHEMBL29404958 0.78 METAP1 (0.56) METAP1ACHE
SCHEMBL20951374 0.78 METAP1 (0.53) METAP1PBRM1TDP2PARP10PARP11
SCHEMBL29594656 0.78 METAP1 (0.53) METAP1PBRM1TDP2PARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed